Compile Data Set for Download or QSAR

Found 70 hits of Enzyme Inhibition Constant Data   

TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361851(CHEMBL1938803 | US9150577, 55)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360292(CHEMBL1933279 | US9150577, 64)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360288(CHEMBL1933148 | US9150577, 23)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360282(CHEMBL1933143 | US9150577, 193)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361841(CHEMBL1938786 | US9150577, 215)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361845(CHEMBL1938792 | US9150577, 108)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361842(CHEMBL1938787 | US9150577, 156)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361847(CHEMBL1938798 | US9150577, 190)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361835(CHEMBL1938765 | US9150577, 10)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361846(CHEMBL1938794 | US9150577, 15)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361839(CHEMBL1938776)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361867(CHEMBL1938791 | US9150577, 226)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361848(CHEMBL1938799 | US9150577, 19)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361849(CHEMBL1938800 | US9150577, 5)copy SMILEScopy InChI
Affinity DataIC50: 68nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361870(CHEMBL1938796)copy SMILEScopy InChI
Affinity DataIC50: 93nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361837(CHEMBL1938774)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361873(CHEMBL1938782 | US9150577, 4)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360282(CHEMBL1933143 | US9150577, 193)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of RSK2-mediated CREB phosphorylation in HeLa cells expressing luciferase reporter geneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360292(CHEMBL1933279 | US9150577, 64)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of RSK2-mediated CREB phosphorylation in HeLa cells expressing luciferase reporter geneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361838(CHEMBL1938775)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361843(CHEMBL1938788 | US9150577, 154)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361853(CHEMBL1938766)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM30298(indole-based 7-membered lactam, 23a)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361874(CHEMBL1938783 | US9150577, 1)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361845(CHEMBL1938792 | US9150577, 108)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Inhibition of RSK2-mediated CREB phosphorylation in HeLa cells expressing luciferase reporter geneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361840(CHEMBL1938781 | US9150577, 178)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361847(CHEMBL1938798 | US9150577, 190)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibition of RSK2-mediated CREB phosphorylation in HeLa cells expressing luciferase reporter geneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361862(CHEMBL257321)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361850(CHEMBL1938802 | US9150577, 112)copy SMILEScopy InChI
Affinity DataIC50: 367nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361865(CHEMBL1938785 | US9150577, 147)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361857(CHEMBL1938770 | US9150577, 123)copy SMILEScopy InChI
Affinity DataIC50: 410nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361869(CHEMBL1938795 | US9150577, 11)copy SMILEScopy InChI
Affinity DataIC50: 540nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361841(CHEMBL1938786 | US9150577, 215)copy SMILEScopy InChI
Affinity DataIC50: 560nMAssay Description:Inhibition of RSK2-mediated CREB phosphorylation in HeLa cells expressing luciferase reporter geneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361842(CHEMBL1938787 | US9150577, 156)copy SMILEScopy InChI
Affinity DataIC50: 620nMAssay Description:Inhibition of RSK2-mediated CREB phosphorylation in HeLa cells expressing luciferase reporter geneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM30283(indole-based 6-membered lactam, 2)copy SMILEScopy InChI
Affinity DataIC50: 730nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360288(CHEMBL1933148 | US9150577, 23)copy SMILEScopy InChI
Affinity DataIC50: 790nMAssay Description:Inhibition of RSK2-mediated CREB phosphorylation in HeLa cells expressing luciferase reporter geneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361839(CHEMBL1938776)copy SMILEScopy InChI
Affinity DataIC50: 840nMAssay Description:Inhibition of RSK2-mediated CREB phosphorylation in HeLa cells expressing luciferase reporter geneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361848(CHEMBL1938799 | US9150577, 19)copy SMILEScopy InChI
Affinity DataIC50: 840nMAssay Description:Inhibition of RSK2-mediated CREB phosphorylation in HeLa cells expressing luciferase reporter geneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361861(CHEMBL1938777)copy SMILEScopy InChI
Affinity DataIC50: 871nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361835(CHEMBL1938765 | US9150577, 10)copy SMILEScopy InChI
Affinity DataIC50: 890nMAssay Description:Inhibition of RSK2-mediated CREB phosphorylation in HeLa cells expressing luciferase reporter geneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM30284(indole-based 6-membered lactam, (R)-4a)copy SMILEScopy InChI
Affinity DataIC50: 970nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361871(CHEMBL1938797)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361854(CHEMBL1938767 | US9150577, 151)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361849(CHEMBL1938800 | US9150577, 5)copy SMILEScopy InChI
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of RSK2-mediated CREB phosphorylation in HeLa cells expressing luciferase reporter geneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361836(CHEMBL272096)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361838(CHEMBL1938775)copy SMILEScopy InChI
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of RSK2-mediated CREB phosphorylation in HeLa cells expressing luciferase reporter geneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361837(CHEMBL1938774)copy SMILEScopy InChI
Affinity DataIC50: 1.63E+3nMAssay Description:Inhibition of RSK2-mediated CREB phosphorylation in HeLa cells expressing luciferase reporter geneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361856(CHEMBL1938769 | US9150577, 152)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361852(CHEMBL272309)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50361840(CHEMBL1938781 | US9150577, 178)copy SMILEScopy InChI
Affinity DataIC50: 1.93E+3nMAssay Description:Inhibition of RSK2-mediated CREB phosphorylation in HeLa cells expressing luciferase reporter geneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
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