Found 32 hits of Enzyme Inhibition Constant Data
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 113nMAssay Description:Inhibition of wild type EGFR using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation cou...More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of wild type B-Raf using MEK1-KM as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 399nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 8.20E+4nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 8.70E+4nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of VEGFR2 using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Islamic University of Gaza
Curated by ChEMBL
Islamic University of Gaza
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SRC using poly(Glu,Tyr) as substrate assessed as [33P-gamma]-ATP incorporation after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
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