Compile Data Set for Download or QSAR

Found 55 hits of Enzyme Inhibition Constant Data   

TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364748(CHEMBL1952100)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364751(CHEMBL1951908)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364745(CHEMBL1951916)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364743(CHEMBL1951914)copy SMILEScopy InChI
Affinity DataIC50: 0.260nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50185666((R)-N-(1-(3-(3,5-difluorophenyl)-3-(4-(methylsulfo...)copy SMILEScopy InChI
Affinity DataIC50: 0.320nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364771(CHEMBL1951913)copy SMILEScopy InChI
Affinity DataIC50: 0.440nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364746(CHEMBL1951917)copy SMILEScopy InChI
Affinity DataIC50: 0.550nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364770(CHEMBL1951912)copy SMILEScopy InChI
Affinity DataIC50: 0.680nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364743(CHEMBL1951914)copy SMILEScopy InChI
Affinity DataIC50: 0.690nMAssay Description:Antagonist activity at CCR5 in allo T cells assessed as inhibition of MIP-1beta-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364744(CHEMBL1951915)copy SMILEScopy InChI
Affinity DataIC50: 0.690nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364750(CHEMBL1951906)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364752(CHEMBL1951898)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364766(CHEMBL1951907)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364756(CHEMBL1951894)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364747(CHEMBL1951918)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364769(CHEMBL1951911)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364755(CHEMBL1951893)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364767(CHEMBL1949696)copy SMILEScopy InChI
Affinity DataIC50: 5.40nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364764(CHEMBL1951904)copy SMILEScopy InChI
Affinity DataIC50: 8.90nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364753(CHEMBL1951899)copy SMILEScopy InChI
Affinity DataIC50: 8.90nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364759(CHEMBL1951897)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364749(CHEMBL1951909)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Displacement of 3,7-Bis[2-(4-nitro[3,5-3H]phenyl)ethyl]-3,7-diazabicyclo[3.3.1]nonane from human ERG expressed in HEK cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364765(CHEMBL1951905)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364758(CHEMBL1951896)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364762(CHEMBL1951902)copy SMILEScopy InChI
Affinity DataIC50: 83nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364763(CHEMBL1951903)copy SMILEScopy InChI
Affinity DataIC50: 126nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364761(CHEMBL1951901)copy SMILEScopy InChI
Affinity DataIC50: 162nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364757(CHEMBL1951895)copy SMILEScopy InChI
Affinity DataIC50: 229nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364760(CHEMBL1951900)copy SMILEScopy InChI
Affinity DataIC50: 339nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364754(CHEMBL1951892)copy SMILEScopy InChI
Affinity DataIC50: 363nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364768(CHEMBL1951910)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364751(CHEMBL1951908)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of 3,7-Bis[2-(4-nitro[3,5-3H]phenyl)ethyl]-3,7-diazabicyclo[3.3.1]nonane from human ERG expressed in HEK cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50185666((R)-N-(1-(3-(3,5-difluorophenyl)-3-(4-(methylsulfo...)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human ERG by electrophysiological assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364756(CHEMBL1951894)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+3nMAssay Description:Displacement of 3,7-Bis[2-(4-nitro[3,5-3H]phenyl)ethyl]-3,7-diazabicyclo[3.3.1]nonane from human ERG expressed in HEK cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364752(CHEMBL1951898)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+3nMAssay Description:Displacement of 3,7-Bis[2-(4-nitro[3,5-3H]phenyl)ethyl]-3,7-diazabicyclo[3.3.1]nonane from human ERG expressed in HEK cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364749(CHEMBL1951909)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364745(CHEMBL1951916)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMAssay Description:Displacement of 3,7-Bis[2-(4-nitro[3,5-3H]phenyl)ethyl]-3,7-diazabicyclo[3.3.1]nonane from human ERG expressed in HEK cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364753(CHEMBL1951899)copy SMILEScopy InChI
Affinity DataIC50: 5.80E+3nMAssay Description:Displacement of 3,7-Bis[2-(4-nitro[3,5-3H]phenyl)ethyl]-3,7-diazabicyclo[3.3.1]nonane from human ERG expressed in HEK cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364748(CHEMBL1952100)copy SMILEScopy InChI
Affinity DataIC50: 6.50E+3nMAssay Description:Displacement of 3,7-Bis[2-(4-nitro[3,5-3H]phenyl)ethyl]-3,7-diazabicyclo[3.3.1]nonane from human ERG expressed in HEK cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50185666((R)-N-(1-(3-(3,5-difluorophenyl)-3-(4-(methylsulfo...)copy SMILEScopy InChI
Affinity DataIC50: 7.30E+3nMAssay Description:Displacement of 3,7-Bis[2-(4-nitro[3,5-3H]phenyl)ethyl]-3,7-diazabicyclo[3.3.1]nonane from human ERG expressed in HEK cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364747(CHEMBL1951918)copy SMILEScopy InChI
Affinity DataIC50: 7.90E+3nMAssay Description:Displacement of 3,7-Bis[2-(4-nitro[3,5-3H]phenyl)ethyl]-3,7-diazabicyclo[3.3.1]nonane from human ERG expressed in HEK cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364746(CHEMBL1951917)copy SMILEScopy InChI
Affinity DataIC50: 7.90E+3nMAssay Description:Displacement of 3,7-Bis[2-(4-nitro[3,5-3H]phenyl)ethyl]-3,7-diazabicyclo[3.3.1]nonane from human ERG expressed in HEK cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364743(CHEMBL1951914)copy SMILEScopy InChI
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364743(CHEMBL1951914)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human ERG by electrophysiological assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364755(CHEMBL1951893)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Displacement of 3,7-Bis[2-(4-nitro[3,5-3H]phenyl)ethyl]-3,7-diazabicyclo[3.3.1]nonane from human ERG expressed in HEK cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364744(CHEMBL1951915)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+4nMAssay Description:Displacement of 3,7-Bis[2-(4-nitro[3,5-3H]phenyl)ethyl]-3,7-diazabicyclo[3.3.1]nonane from human ERG expressed in HEK cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364743(CHEMBL1951914)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364743(CHEMBL1951914)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+4nMAssay Description:Displacement of 3,7-Bis[2-(4-nitro[3,5-3H]phenyl)ethyl]-3,7-diazabicyclo[3.3.1]nonane from human ERG expressed in HEK cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364758(CHEMBL1951896)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+4nMAssay Description:Displacement of 3,7-Bis[2-(4-nitro[3,5-3H]phenyl)ethyl]-3,7-diazabicyclo[3.3.1]nonane from human ERG expressed in HEK cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50364750(CHEMBL1951906)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+4nMAssay Description:Displacement of 3,7-Bis[2-(4-nitro[3,5-3H]phenyl)ethyl]-3,7-diazabicyclo[3.3.1]nonane from human ERG expressed in HEK cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GQ6PubMed
Displayed 1 to 50 (of 55 total ) | Next | Last >>* indicates data uncertainty>20%