Compile Data Set for Download or QSAR

Found 116 hits of Enzyme Inhibition Constant Data   

TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389695(CHEMBL2070062 | US10544104, Compound 40 | US112479...)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345740(3-(6-ethoxynaphthalen-2-yl)-1-isopropyl-1H-pyrazol...)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Inhibition of human LCK using Ac-EIYGEFKKK-OH as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345738(1-isopropyl-3-(naphthalen-2-yl)-1H-pyrazolo[3,4-d]...)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345739(1-isopropyl-3-(6-methoxynaphthalen-2-yl)-1H-pyrazo...)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibition of human LCK using Ac-EIYGEFKKK-OH as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389703(CHEMBL2070075 | US10544104, Compound 148 | US97650...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of human LCK using Ac-EIYGEFKKK-OH as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345704(1-(tert-butyl)-3-(naphthalen-2-yl)-1H-pyrazolo[3,4...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM123747(1-(tert-butyl)-3-phenyl-1H-pyrazolo[3,4-d]pyrimidi...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389728(CHEMBL2069944 | US10544104, Compound 132 | US97650...)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345742(1-isopropyl-3-(quinolin-3-yl)-1H-pyrazolo[3,4-d]py...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389687(CHEMBL2070054 | US10544104, Compound 41 | US112479...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389691(CHEMBL2070057 | US10544104, Compound 43 | US112479...)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389701(CHEMBL2070068 | US10544104, Compound 56 | US112479...)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389697(CHEMBL2070064 | US10544104, Compound 46 | US112479...)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389699(CHEMBL2070066 | US10544104, Compound 47 | US112479...)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389734(CHEMBL2069950 | US10544104, Compound 20 | US112479...)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389689(CHEMBL2070055 | US10544104, Compound 12 | US112479...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345740(3-(6-ethoxynaphthalen-2-yl)-1-isopropyl-1H-pyrazol...)copy SMILEScopy InChI
Affinity DataIC50: 380nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389700(CHEMBL2070067 | US10544104, Compound 38 | US112479...)copy SMILEScopy InChI
Affinity DataIC50: 380nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345739(1-isopropyl-3-(6-methoxynaphthalen-2-yl)-1H-pyrazo...)copy SMILEScopy InChI
Affinity DataIC50: 510nMAssay Description:Inhibition of human EGFR using poly glu-Tyr as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389735(CHEMBL2069951 | US10544104, Compound 139 | US97650...)copy SMILEScopy InChI
Affinity DataIC50: 520nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389685(CHEMBL2070052 | US10544104, Compound 11 | US112479...)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389725(CHEMBL2069941 | US10544104, Compound 134 | US97650...)copy SMILEScopy InChI
Affinity DataIC50: 580nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50383380(CHEMBL2030553 | CHEMBL2070047 | US10544104, Compou...)copy SMILEScopy InChI
Affinity DataIC50: 620nMAssay Description:Inhibition of human LCK using Ac-EIYGEFKKK-OH as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345735(1-isopropyl-3-(4-methoxy-3-methylphenyl)-1H-pyrazo...)copy SMILEScopy InChI
Affinity DataIC50: 650nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345739(1-isopropyl-3-(6-methoxynaphthalen-2-yl)-1H-pyrazo...)copy SMILEScopy InChI
Affinity DataIC50: 670nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345740(3-(6-ethoxynaphthalen-2-yl)-1-isopropyl-1H-pyrazol...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Inhibition of human EGFR using poly glu-Tyr as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389711(CHEMBL2070078 | US10307425, Example 113 | US106321...)copy SMILEScopy InChI
Affinity DataIC50: 730nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389694(CHEMBL2070060 | US10544104, Compound 42 | US112479...)copy SMILEScopy InChI
Affinity DataIC50: 780nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389713(CHEMBL2070080)copy SMILEScopy InChI
Affinity DataIC50: 810nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345739(1-isopropyl-3-(6-methoxynaphthalen-2-yl)-1H-pyrazo...)copy SMILEScopy InChI
Affinity DataIC50: 820nMAssay Description:Inhibition of human ABL using EAIYAAPFAKKK-OH as substrate by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50383381(CHEMBL2030554 | CHEMBL2070050 | US10544104, Compou...)copy SMILEScopy InChI
Affinity DataIC50: 960nMAssay Description:Inhibition of human LCK using Ac-EIYGEFKKK-OH as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389692(CHEMBL2070058)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50383382(CHEMBL2030556 | CHEMBL2069948 | US10172858, Table ...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345729(1-isopropyl-3-m-tolyl-1H-pyrazolo[3,4-d]pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389730(CHEMBL2069946 | US10172858, Table 2.7 | US10544104...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetEphrin type-A receptor 3(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345739(1-isopropyl-3-(6-methoxynaphthalen-2-yl)-1H-pyrazo...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human EPHA3 using myelin basic protein as substrate after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389702(CHEMBL2070069 | US10544104, Compound 39 | US112479...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389712(CHEMBL2070079)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345740(3-(6-ethoxynaphthalen-2-yl)-1-isopropyl-1H-pyrazol...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human ABL using EAIYAAPFAKKK-OH as substrate by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389698(CHEMBL2070065 | US10544104, Compound 37 | US112479...)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389679(CHEMBL2070046 | US10544104, Compound 135 | US97650...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389736(CHEMBL2069952 | US10544104, Compound 142 | US97650...)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50298225(CHEMBL2069955 | CHEMBL573578 | NM-PP1 | US10544104...)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389682(CHEMBL2070049 | US10544104, Compound 137 | US95180...)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345739(1-isopropyl-3-(6-methoxynaphthalen-2-yl)-1H-pyrazo...)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human CSK using Ac-KKKKEEIYFFF-OH as substrate after 180 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389696(CHEMBL2070063 | US10544104, Compound 34 | US112479...)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345740(3-(6-ethoxynaphthalen-2-yl)-1-isopropyl-1H-pyrazol...)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human CSK using Ac-KKKKEEIYFFF-OH as substrate after 180 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389717(CHEMBL2070085 | US10307425, Example 107 | US106321...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389704(CHEMBL2070081 | US10544104, Compound 150 | US95180...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human LCK using Ac-EIYGEFKKK-OH as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetEphrin type-A receptor 3(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50345740(3-(6-ethoxynaphthalen-2-yl)-1-isopropyl-1H-pyrazol...)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of human EPHA3 using myelin basic protein as substrate after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
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