Compile Data Set for Download or QSAR

Found 82 hits of Enzyme Inhibition Constant Data   

TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381179(CHEMBL2018388)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381182(CHEMBL2018391)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381174(CHEMBL2018380)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381177(CHEMBL2018386)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381188(CHEMBL2018400)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381181(CHEMBL2018390)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381175(CHEMBL2018384)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381177(CHEMBL2018386)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Antagonist activity at CCR2 in mouse monocytes assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381179(CHEMBL2018388)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381190(CHEMBL2018402)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381178(CHEMBL2018387)copy SMILEScopy InChI
Affinity DataIC50: 4.70nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381173(CHEMBL2018370)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381201(CHEMBL2018371)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381176(CHEMBL2018385)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381180(CHEMBL2018389)copy SMILEScopy InChI
Affinity DataIC50: 5.20nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381183(CHEMBL2018392)copy SMILEScopy InChI
Affinity DataIC50: 5.30nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381180(CHEMBL2018389)copy SMILEScopy InChI
Affinity DataIC50: 5.80nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381176(CHEMBL2018385)copy SMILEScopy InChI
Affinity DataIC50: 6.70nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381167(CHEMBL2018396)copy SMILEScopy InChI
Affinity DataIC50: 6.70nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381209(CHEMBL2018381)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381189(CHEMBL2018401)copy SMILEScopy InChI
Affinity DataIC50: 7.10nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381185(CHEMBL2018394)copy SMILEScopy InChI
Affinity DataIC50: 7.20nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381184(CHEMBL2018393)copy SMILEScopy InChI
Affinity DataIC50: 7.40nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381183(CHEMBL2018392)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381185(CHEMBL2018394)copy SMILEScopy InChI
Affinity DataIC50: 9.30nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381178(CHEMBL2018387)copy SMILEScopy InChI
Affinity DataIC50: 9.90nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381182(CHEMBL2018391)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381186(CHEMBL2018395)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381169(CHEMBL2018538)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381190(CHEMBL2018402)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381181(CHEMBL2018390)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381188(CHEMBL2018400)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381175(CHEMBL2018384)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381207(CHEMBL2018378)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381203(CHEMBL2018373)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381204(CHEMBL2018374)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381214(CHEMBL2018403)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381167(CHEMBL2018396)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381189(CHEMBL2018401)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381191(CHEMBL2018530)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381177(CHEMBL2018386)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381191(CHEMBL2018530)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381210(CHEMBL2018382)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381187(CHEMBL2018397)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381193(CHEMBL2018363)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381174(CHEMBL2018380)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381184(CHEMBL2018393)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381216(CHEMBL2018528)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381208(CHEMBL2018379)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50381212(CHEMBL2018398)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Displacement of [125-I]MCP1 from CCR2 on human PBMCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN96MBPubMed
Displayed 1 to 50 (of 82 total ) | Next | Last >>* indicates data uncertainty>20%