Compile Data Set for Download or QSAR

Found 210 hits of Enzyme Inhibition Constant Data   

LigandPNGBDBM50393357(CHEMBL2152148)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393365(CHEMBL2152257)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393359(CHEMBL2152150)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393333(CHEMBL2151050)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393348(CHEMBL2152139)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393339(CHEMBL2152131)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393360(CHEMBL2152250)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393342(CHEMBL2152252)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
LigandPNGBDBM50393335(CHEMBL2152127)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393353(CHEMBL2152144)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393334(CHEMBL2152126)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
LigandPNGBDBM50393364(CHEMBL2152256)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393354(CHEMBL2152145)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393332(CHEMBL2152125)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
LigandPNGBDBM50393358(CHEMBL2152149)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393340(CHEMBL2152132)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393355(CHEMBL2152146)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393351(CHEMBL2152142)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393329(CHEMBL2152253)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393333(CHEMBL2151050)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of human PI3Kalpha expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393365(CHEMBL2152257)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of human PI3Kbeta expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescenc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393338(CHEMBL2152130)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393365(CHEMBL2152257)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of human PI3Kdelta expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393356(CHEMBL2152147)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
LigandPNGBDBM50393350(CHEMBL2152141)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393349(CHEMBL2152140)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393352(CHEMBL2152143)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393345(CHEMBL2152136)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393364(CHEMBL2152256)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Inhibition of human PI3Kbeta expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescenc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393337(CHEMBL2152129)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393363(CHEMBL2152255)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393348(CHEMBL2152139)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of human PI3Kbeta expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescenc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393341(CHEMBL2152133)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393338(CHEMBL2152130)copy SMILEScopy InChI
Affinity DataIC50: 69nMAssay Description:Inhibition of human PI3Kgamma expressed in C5a-stimulated mouse RAW 264.7 cells assessed as inhibition of AKT phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393348(CHEMBL2152139)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of human PI3Kalpha expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393340(CHEMBL2152132)copy SMILEScopy InChI
Affinity DataIC50: 97nMAssay Description:Inhibition of human PI3Kalpha expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393348(CHEMBL2152139)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of human PI3Kdelta expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393361(CHEMBL2152251)copy SMILEScopy InChI
Affinity DataIC50: 102nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393365(CHEMBL2152257)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of human PI3Kalpha expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393355(CHEMBL2152146)copy SMILEScopy InChI
Affinity DataIC50: 142nMAssay Description:Inhibition of human PI3Kalpha expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393339(CHEMBL2152131)copy SMILEScopy InChI
Affinity DataIC50: 142nMAssay Description:Inhibition of human PI3Kalpha expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393344(CHEMBL2152135)copy SMILEScopy InChI
Affinity DataIC50: 152nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393347(CHEMBL2152138)copy SMILEScopy InChI
Affinity DataIC50: 161nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393346(CHEMBL2152137)copy SMILEScopy InChI
Affinity DataIC50: 167nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393350(CHEMBL2152141)copy SMILEScopy InChI
Affinity DataIC50: 171nMAssay Description:Inhibition of human PI3Kgamma expressed in C5a-stimulated mouse RAW 264.7 cells assessed as inhibition of AKT phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393338(CHEMBL2152130)copy SMILEScopy InChI
Affinity DataIC50: 174nMAssay Description:Inhibition of human PI3Kalpha expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393353(CHEMBL2152144)copy SMILEScopy InChI
Affinity DataIC50: 174nMAssay Description:Inhibition of human PI3Kalpha expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393364(CHEMBL2152256)copy SMILEScopy InChI
Affinity DataIC50: 181nMAssay Description:Inhibition of human PI3Kdelta expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6S9NPubMed
LigandPNGBDBM50393334(CHEMBL2152126)copy SMILEScopy InChI
Affinity DataIC50: 182nMAssay Description:Inhibition of human PI3Kgamma expressed in C5a-stimulated mouse RAW 264.7 cells assessed as inhibition of AKT phosphorylation by ELISAMore data for this Ligand-Target Pair
Displayed 1 to 50 (of 210 total ) | Next | Last >>* indicates data uncertainty>20%