Found 11 hits of Enzyme Inhibition Constant Data
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
National Center for Advancing Translation Sciences
Curated by ChEMBL
National Center for Advancing Translation Sciences
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of wild type glucocerebrosidase using 4-methylumbellifereno-Glc as substrate incubated for 5 mins prior to substrate addition measured aft...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
National Center for Advancing Translation Sciences
Curated by ChEMBL
National Center for Advancing Translation Sciences
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of wild type glucocerebrosidase using 4-methylumbellifereno-Glc as substrate incubated for 5 mins prior to substrate addition measured aft...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
National Center for Advancing Translation Sciences
Curated by ChEMBL
National Center for Advancing Translation Sciences
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of wild type glucocerebrosidase using 4-methylumbellifereno-Glc as substrate incubated for 5 mins prior to substrate addition measured aft...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
National Center for Advancing Translation Sciences
Curated by ChEMBL
National Center for Advancing Translation Sciences
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of wild type glucocerebrosidase in human spleen homogenate using 4-methylumbellifereno-Glc as substrate incubated for 5 mins prior to subs...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
National Center for Advancing Translation Sciences
Curated by ChEMBL
National Center for Advancing Translation Sciences
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of wild type glucocerebrosidase in human spleen homogenate using 4-methylumbellifereno-Glc as substrate incubated for 5 mins prior to subs...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
National Center for Advancing Translation Sciences
Curated by ChEMBL
National Center for Advancing Translation Sciences
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of wild type glucocerebrosidase using 4-methylumbellifereno-Glc as substrate incubated for 5 mins prior to substrate addition measured aft...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
National Center for Advancing Translation Sciences
Curated by ChEMBL
National Center for Advancing Translation Sciences
Curated by ChEMBL
Affinity DataIC50: 710nMAssay Description:Inhibition of wild type glucocerebrosidase using 4-methylumbellifereno-Glc as substrate incubated for 5 mins prior to substrate addition measured aft...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
National Center for Advancing Translation Sciences
Curated by ChEMBL
National Center for Advancing Translation Sciences
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of wild type glucocerebrosidase in human spleen homogenate using 4-methylumbellifereno-Glc as substrate incubated for 5 mins prior to subs...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
National Center for Advancing Translation Sciences
Curated by ChEMBL
National Center for Advancing Translation Sciences
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of wild type glucocerebrosidase in human spleen homogenate using 4-methylumbellifereno-Glc as substrate incubated for 5 mins prior to subs...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
National Center for Advancing Translation Sciences
Curated by ChEMBL
National Center for Advancing Translation Sciences
Curated by ChEMBL
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of wild type glucocerebrosidase in human spleen homogenate using 4-methylumbellifereno-Glc as substrate incubated for 5 mins prior to subs...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
National Center for Advancing Translation Sciences
Curated by ChEMBL
National Center for Advancing Translation Sciences
Curated by ChEMBL
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of wild type glucocerebrosidase using 4-methylumbellifereno-Glc as substrate incubated for 5 mins prior to substrate addition measured aft...More data for this Ligand-Target Pair