Compile Data Set for Download or QSAR

Found 4 hits of Enzyme Inhibition Constant Data   

TargetGlucagon receptor(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50396184(REDIOCIDE A)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of GCGR expressed in HEK293 cells assessed as inhibition of calcium influx after 10 mins by Fluo-4-AM based fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7PW9PubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50396184(REDIOCIDE A)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of adrenergic receptor 1a expressed in HEK293 cells assessed as inhibition of calcium influx after 10 mins by Fluo-4-AM based fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7PW9PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50396184(REDIOCIDE A)copy SMILEScopy InChI
Affinity DataIC50: 215nMAssay Description:Inhibition of adrenergic receptor 1b receptor expressed in HEK293 cells assessed as inhibition of calcium influx after 10 mins by Fluo-4-AM based flu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7PW9PubMed
TargetC-C chemokine receptor type 6(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50396184(REDIOCIDE A)copy SMILEScopy InChI
Affinity DataIC50: 261nMAssay Description:Inhibition of CCR6 expressed in HEK293 cells assessed as inhibition of calcium influx after 10 mins by Fluo-4-AM based fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7PW9PubMed
* indicates data uncertainty>20%