Compile Data Set for Download or QSAR

Found 12 hits of Enzyme Inhibition Constant Data   

TargetTyrosine-protein kinase HCK(Homo sapiens (Human))
University of Washington

LigandPNGBDBM93207(Kinase inhibitor, 5)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMpH: 7.5 T: 2°CAssay Description:Fluorescence assay used for determination of catch and release efficiency. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9N1XPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

LigandPNGBDBM93207(Kinase inhibitor, 5)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:Fluorescence assay used for determination of catch and release efficiency. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9N1XPubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University of Washington

LigandPNGBDBM93207(Kinase inhibitor, 5)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:Fluorescence assay used for determination of catch and release efficiency. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9N1XPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Washington

LigandPNGBDBM93207(Kinase inhibitor, 5)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:Fluorescence assay used for determination of catch and release efficiency. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9N1XPubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University of Washington

LigandPNGBDBM93207(Kinase inhibitor, 5)copy SMILEScopy InChI
Affinity DataIC50: 8.40nMpH: 7.5 T: 2°CAssay Description:Fluorescence assay used for determination of catch and release efficiency. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9N1XPubMed
TargetSerine/threonine-protein kinase 10(Homo sapiens (Human))
University of Washington

LigandPNGBDBM93207(Kinase inhibitor, 5)copy SMILEScopy InChI
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:Fluorescence assay used for determination of catch and release efficiency. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9N1XPubMed
TargetEphrin type-A receptor 3(Homo sapiens (Human))
University of Washington

LigandPNGBDBM93207(Kinase inhibitor, 5)copy SMILEScopy InChI
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:Fluorescence assay used for determination of catch and release efficiency. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9N1XPubMed
TargetSerine/threonine-protein kinase 10(Homo sapiens (Human))
University of Washington

LigandPNGBDBM93207(Kinase inhibitor, 5)copy SMILEScopy InChI
Affinity DataIC50: 20nMpH: 7.5 T: 2°CAssay Description:Fluorescence assay used for determination of catch and release efficiency. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9N1XPubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
University of Washington

LigandPNGBDBM93207(Kinase inhibitor, 5)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Fluorescence assay used for determination of catch and release efficiency. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9N1XPubMed
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
University of Washington

LigandPNGBDBM93207(Kinase inhibitor, 5)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Fluorescence assay used for determination of catch and release efficiency. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9N1XPubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
University of Washington

LigandPNGBDBM93207(Kinase inhibitor, 5)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Fluorescence assay used for determination of catch and release efficiency. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9N1XPubMed
TargetSerine/threonine-protein kinase PAK 5(Homo sapiens (Human))
University of Washington

LigandPNGBDBM93207(Kinase inhibitor, 5)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Fluorescence assay used for determination of catch and release efficiency. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9N1XPubMed
* indicates data uncertainty>20%