Compile Data Set for Download or QSAR

Found 166 hits of Enzyme Inhibition Constant Data   

TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490612(CHEMBL2337603)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490637(CHEMBL2338049)copy SMILEScopy InChI
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490602(CHEMBL2338047)copy SMILEScopy InChI
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490621(CHEMBL2338048)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490599(CHEMBL2337596)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490592(CHEMBL2337595)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490625(CHEMBL2338034)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490611(CHEMBL2337604)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490600(CHEMBL2337602)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490606(CHEMBL2338039)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490635(CHEMBL2337593)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490638(CHEMBL2338051)copy SMILEScopy InChI
Affinity DataKi:  63nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490609(CHEMBL2338032)copy SMILEScopy InChI
Affinity DataKi:  63nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490631(CHEMBL2338050)copy SMILEScopy InChI
Affinity DataKi:  63nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490601(CHEMBL2337592)copy SMILEScopy InChI
Affinity DataKi:  63nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490590(CHEMBL2338053)copy SMILEScopy InChI
Affinity DataKi:  79nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490604(CHEMBL2338042)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490624(CHEMBL2338035)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490620(CHEMBL2338054)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490632(CHEMBL2338045)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490633(CHEMBL2338033)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490593(CHEMBL2338043)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490619(CHEMBL2338055)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490630(CHEMBL2338052)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490607(CHEMBL2338037)copy SMILEScopy InChI
Affinity DataKi:  126nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490613(CHEMBL2337598)copy SMILEScopy InChI
Affinity DataKi:  126nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490615(CHEMBL2337594)copy SMILEScopy InChI
Affinity DataKi:  126nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490622(CHEMBL2338044)copy SMILEScopy InChI
Affinity DataKi:  126nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490595(CHEMBL2337605)copy SMILEScopy InChI
Affinity DataKi:  126nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490597(CHEMBL2337591)copy SMILEScopy InChI
Affinity DataKi:  126nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490591(CHEMBL2337590)copy SMILEScopy InChI
Affinity DataKi:  158nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490626(CHEMBL2337608)copy SMILEScopy InChI
Affinity DataKi:  158nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490610(CHEMBL2338031)copy SMILEScopy InChI
Affinity DataKi:  158nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490614(CHEMBL2337597)copy SMILEScopy InChI
Affinity DataKi:  158nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490616(CHEMBL2337589)copy SMILEScopy InChI
Affinity DataKi:  251nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490603(CHEMBL2338046)copy SMILEScopy InChI
Affinity DataKi:  316nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490629(CHEMBL2337606)copy SMILEScopy InChI
Affinity DataKi:  316nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM84745(CAS_136434-34-9 | DULOXETINE | LY-248686 | LY24868...)copy SMILEScopy InChI
Affinity DataKi:  316nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMedDrugBank
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490627(CHEMBL2337607)copy SMILEScopy InChI
Affinity DataKi:  316nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490605(CHEMBL2338041)copy SMILEScopy InChI
Affinity DataKi:  398nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490608(CHEMBL2338036)copy SMILEScopy InChI
Affinity DataKi:  398nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490617(CHEMBL2337587)copy SMILEScopy InChI
Affinity DataKi:  501nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490623(CHEMBL2338040)copy SMILEScopy InChI
Affinity DataKi:  794nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490628(CHEMBL2337586)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490634(CHEMBL2337588)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490598(CHEMBL2338038)copy SMILEScopy InChI
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM35226((S,S)-reboxetine | Reboxetine | Vestra)copy SMILEScopy InChI
Affinity DataKi:  2.00E+4nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490618(Midalcipran | Milnacipran)copy SMILEScopy InChI
Affinity DataKi: <3.16E+4nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM50490621(CHEMBL2338048)copy SMILEScopy InChI
Affinity DataIC50: 0.316nMAssay Description:Inhibition of human recombinant NET expressed in HEK293 cells assessed as inhibition of [3H]NE reuptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Theravance, Inc.

Curated by ChEMBL
LigandPNGBDBM84745(CAS_136434-34-9 | DULOXETINE | LY-248686 | LY24868...)copy SMILEScopy InChI
Affinity DataIC50: 0.316nMAssay Description:Inhibition of human recombinant SERT expressed in HEK293 cells assessed as inhibition of [3H]5HT reuptakeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD14M7PubMedDrugBank
Displayed 1 to 50 (of 166 total ) | Next | Last >>* indicates data uncertainty>20%