Compile Data Set for Download or QSAR

Found 6 hits of Enzyme Inhibition Constant Data   

TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)copy SMILEScopy InChI
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum homogenate after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZMWPubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50448210(CHEMBL3120697 | US9018213, 15)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum homogenate after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZMWPubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50448208(CHEMBL3120688)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum homogenate after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZMWPubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50001885((risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-...)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum homogenate after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZMWPubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50448209(CHEMBL3120682)copy SMILEScopy InChI
Affinity DataKi:  699nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum homogenate after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZMWPubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50448211(CHEMBL3120696)copy SMILEScopy InChI
Affinity DataKi:  1.83E+3nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum homogenate after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZMWPubMed
* indicates data uncertainty>20%