Found 3 hits of Enzyme Inhibition Constant Data
TargetCytochrome P450 2D4(Rattus norvegicus)
Division of Medicinal& Process Chemistry, Division of Parasitology, Division of Pharmacokinetics and Metabolism, and Sophisticated Analytical Instrument Facility, Central Drug Research Institute
Curated by ChEMBL
Division of Medicinal& Process Chemistry, Division of Parasitology, Division of Pharmacokinetics and Metabolism, and Sophisticated Analytical Instrument Facility, Central Drug Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CYP2D4 in rat liver microsome using dextromethorphan as substrate by HPLC-PDA analysisMore data for this Ligand-Target Pair
TargetCytochrome P450 1A2(Rattus norvegicus)
Division of Medicinal& Process Chemistry, Division of Parasitology, Division of Pharmacokinetics and Metabolism, and Sophisticated Analytical Instrument Facility, Central Drug Research Institute
Curated by ChEMBL
Division of Medicinal& Process Chemistry, Division of Parasitology, Division of Pharmacokinetics and Metabolism, and Sophisticated Analytical Instrument Facility, Central Drug Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CYP1A2 in rat liver microsome using phenacetin as substrate by HPLC-PDA analysisMore data for this Ligand-Target Pair
TargetCytochrome P450 2C11(Rattus norvegicus)
Division of Medicinal& Process Chemistry, Division of Parasitology, Division of Pharmacokinetics and Metabolism, and Sophisticated Analytical Instrument Facility, Central Drug Research Institute
Curated by ChEMBL
Division of Medicinal& Process Chemistry, Division of Parasitology, Division of Pharmacokinetics and Metabolism, and Sophisticated Analytical Instrument Facility, Central Drug Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CYP2C11 in rat liver microsome using diclofenac as substrate by HPLC-PDA analysisMore data for this Ligand-Target Pair