Compile Data Set for Download or QSAR

Found 107 hits of Enzyme Inhibition Constant Data   

Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)copy SMILEScopy InChI
Affinity DataKi:  3.40nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50420342(CHEMBL2089156)copy SMILEScopy InChI
Affinity DataKi:  5.80nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417346(CHEMBL1276220)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417344(CHEMBL1276218)copy SMILEScopy InChI
Affinity DataKi:  7.20nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50419878(CHEMBL1956195)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50493433(CHEMBL2431282)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50419880(CHEMBL1956197)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417346(CHEMBL1276220)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417344(CHEMBL1276218)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50419874(CHEMBL1956192)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50412245(CHEMBL495095)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50027060(2-(2-Cyclopropyl-phenoxymethyl)-4,5-dihydro-1H-imi...)copy SMILEScopy InChI
Affinity DataKi:  35nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417343(CHEMBL1276140)copy SMILEScopy InChI
Affinity DataKi:  35nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50419878(CHEMBL1956195)copy SMILEScopy InChI
Affinity DataKi:  36nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50420341(CHEMBL2089155)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50420342(CHEMBL2089156)copy SMILEScopy InChI
Affinity DataKi:  42nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50420341(CHEMBL2089155)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417345(CHEMBL1276219)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473179(CHEMBL13917)copy SMILEScopy InChI
Affinity DataKi:  49nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50493433(CHEMBL2431282)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417343(CHEMBL1276140)copy SMILEScopy InChI
Affinity DataKi:  52nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50412245(CHEMBL495095)copy SMILEScopy InChI
Affinity DataKi:  58nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50027060(2-(2-Cyclopropyl-phenoxymethyl)-4,5-dihydro-1H-imi...)copy SMILEScopy InChI
Affinity DataKi:  59nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417346(CHEMBL1276220)copy SMILEScopy InChI
Affinity DataKi:  63nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473154(CHEMBL14107)copy SMILEScopy InChI
Affinity DataKi:  71nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417343(CHEMBL1276140)copy SMILEScopy InChI
Affinity DataKi:  71nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473154(CHEMBL14107)copy SMILEScopy InChI
Affinity DataKi:  71nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50493430(CHEMBL2431281)copy SMILEScopy InChI
Affinity DataKi:  78nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50493431(CHEMBL2431280)copy SMILEScopy InChI
Affinity DataKi:  79nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473179(CHEMBL13917)copy SMILEScopy InChI
Affinity DataKi:  79nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417344(CHEMBL1276218)copy SMILEScopy InChI
Affinity DataKi:  79nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50419880(CHEMBL1956197)copy SMILEScopy InChI
Affinity DataKi:  83nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50493430(CHEMBL2431281)copy SMILEScopy InChI
Affinity DataKi:  83nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50412245(CHEMBL495095)copy SMILEScopy InChI
Affinity DataKi:  85nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50493432(CHEMBL2431279)copy SMILEScopy InChI
Affinity DataKi:  95nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417342(CHEMBL1276139)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473154(CHEMBL14107)copy SMILEScopy InChI
Affinity DataKi:  126nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417345(CHEMBL1276219)copy SMILEScopy InChI
Affinity DataKi:  126nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50419874(CHEMBL1956192)copy SMILEScopy InChI
Affinity DataKi:  148nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50493433(CHEMBL2431282)copy SMILEScopy InChI
Affinity DataKi:  148nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417342(CHEMBL1276139)copy SMILEScopy InChI
Affinity DataKi:  178nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50420341(CHEMBL2089155)copy SMILEScopy InChI
Affinity DataKi:  234nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417346(CHEMBL1276220)copy SMILEScopy InChI
Affinity DataKi:  263nMAssay Description:Binding affinity at human alpha2B ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50419878(CHEMBL1956195)copy SMILEScopy InChI
Affinity DataKi:  275nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50420342(CHEMBL2089156)copy SMILEScopy InChI
Affinity DataKi:  275nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50419874(CHEMBL1956192)copy SMILEScopy InChI
Affinity DataKi:  282nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417344(CHEMBL1276218)copy SMILEScopy InChI
Affinity DataKi:  309nMAssay Description:Binding affinity at human alpha2B ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50493431(CHEMBL2431280)copy SMILEScopy InChI
Affinity DataKi:  316nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50412245(CHEMBL495095)copy SMILEScopy InChI
Affinity DataKi:  339nMAssay Description:Binding affinity at human alpha2B ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50420341(CHEMBL2089155)copy SMILEScopy InChI
Affinity DataKi:  339nMAssay Description:Binding affinity at human alpha2B ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Displayed 1 to 50 (of 107 total ) | Next | Last >>* indicates data uncertainty>20%