Compile Data Set for Download or QSAR

Found 19 hits of Enzyme Inhibition Constant Data   

TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019941(CHEMBL3287571)copy SMILEScopy InChI
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human GPR40 expressed in mouse A9 cells by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019940(CHEMBL3287570)copy SMILEScopy InChI
Affinity DataEC50:  11nMAssay Description:Agonist activity at human GPR40 expressed in mouse A9 cells by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019938(CHEMBL3287568)copy SMILEScopy InChI
Affinity DataEC50:  36nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by aequorin assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019971(CHEMBL3287576)copy SMILEScopy InChI
Affinity DataEC50:  57nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by aequorin assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50362690(AMG-837 | CHEMBL1829173)copy SMILEScopy InChI
Affinity DataEC50:  41nMAssay Description:Agonist activity at human GPR40 expressed in mouse A9 cells by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019970(CHEMBL3287575)copy SMILEScopy InChI
Affinity DataEC50:  69nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by aequorin assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019971(CHEMBL3287576)copy SMILEScopy InChI
Affinity DataEC50:  9nMAssay Description:Agonist activity at human GPR40 expressed in mouse A9 cells by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019943(CHEMBL3287572)copy SMILEScopy InChI
Affinity DataEC50:  65nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by aequorin assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019944(CHEMBL3287573)copy SMILEScopy InChI
Affinity DataEC50:  41nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by aequorin assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019969(CHEMBL3287574)copy SMILEScopy InChI
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at human GPR40 expressed in mouse A9 cells by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019939(CHEMBL3287569)copy SMILEScopy InChI
Affinity DataEC50:  33nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by aequorin assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019940(CHEMBL3287570)copy SMILEScopy InChI
Affinity DataEC50:  33nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by aequorin assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019944(CHEMBL3287573)copy SMILEScopy InChI
Affinity DataEC50:  3.80nMAssay Description:Agonist activity at human GPR40 expressed in mouse A9 cells by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019941(CHEMBL3287571)copy SMILEScopy InChI
Affinity DataEC50:  12nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by aequorin assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019942(CHEMBL3286409)copy SMILEScopy InChI
Affinity DataEC50:  73nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by aequorin assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019969(CHEMBL3287574)copy SMILEScopy InChI
Affinity DataEC50:  36nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by aequorin assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019942(CHEMBL3286409)copy SMILEScopy InChI
Affinity DataEC50:  16nMAssay Description:Agonist activity at human GPR40 expressed in mouse A9 cells by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50019939(CHEMBL3287569)copy SMILEScopy InChI
Affinity DataEC50:  7.60nMAssay Description:Agonist activity at human GPR40 expressed in mouse A9 cells by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50362690(AMG-837 | CHEMBL1829173)copy SMILEScopy InChI
Affinity DataEC50:  104nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by aequorin assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028T3MPubMed
* indicates data uncertainty>20%