Compile Data Set for Download or QSAR

Found 36 hits of Enzyme Inhibition Constant Data   

TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102104(CHEMBL3337659)copy SMILEScopy InChI
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102106(CHEMBL3337657)copy SMILEScopy InChI
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50355329(CHEMBL1835336)copy SMILEScopy InChI
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillati...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102172(CHEMBL1835332)copy SMILEScopy InChI
Affinity DataKi:  4.70E+3nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102105(CHEMBL3337658)copy SMILEScopy InChI
Affinity DataKi:  6.30E+3nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102172(CHEMBL1835332)copy SMILEScopy InChI
Affinity DataKi:  1.23E+4nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102171(CHEMBL1835339)copy SMILEScopy InChI
Affinity DataKi:  1.33E+4nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50355329(CHEMBL1835336)copy SMILEScopy InChI
Affinity DataKi:  1.44E+4nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102171(CHEMBL1835339)copy SMILEScopy InChI
Affinity DataKi:  1.70E+4nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102252(CHEMBL3337651)copy SMILEScopy InChI
Affinity DataKi:  1.90E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102107(CHEMBL3337656)copy SMILEScopy InChI
Affinity DataKi:  2.10E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102108(CHEMBL3337650)copy SMILEScopy InChI
Affinity DataKi:  2.40E+4nMAssay Description:Displacement of [3H]SYM2081 from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102108(CHEMBL3337650)copy SMILEScopy InChI
Affinity DataKi:  2.90E+4nMAssay Description:Displacement of [3H]SYM2081 from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102109(CHEMBL3337662)copy SMILEScopy InChI
Affinity DataKi:  3.20E+4nMAssay Description:Displacement of [3H]SYM2081 from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102104(CHEMBL3337659)copy SMILEScopy InChI
Affinity DataKi:  3.40E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102105(CHEMBL3337658)copy SMILEScopy InChI
Affinity DataKi:  4.00E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102107(CHEMBL3337656)copy SMILEScopy InChI
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102250(CHEMBL3337660)copy SMILEScopy InChI
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102170(CHEMBL3358461)copy SMILEScopy InChI
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [3H]SYM2081 from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102106(CHEMBL3337657)copy SMILEScopy InChI
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102109(CHEMBL3337662)copy SMILEScopy InChI
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [3H]SYM2081 from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102252(CHEMBL3337651)copy SMILEScopy InChI
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102250(CHEMBL3337660)copy SMILEScopy InChI
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102110(CHEMBL3358462)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]SYM2081 from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102253(CHEMBL3337652)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102254(CHEMBL3337653)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102280(CHEMBL3337654)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102170(CHEMBL3358461)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]SYM2081 from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102455(CHEMBL3337655)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102110(CHEMBL3358462)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]SYM2081 from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102455(CHEMBL3337655)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102280(CHEMBL3337654)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102237(CHEMBL3337661)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102253(CHEMBL3337652)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102237(CHEMBL3337661)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50102254(CHEMBL3337653)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CXKPubMed
* indicates data uncertainty>20%