Compile Data Set for Download or QSAR

Found 171 hits of Enzyme Inhibition Constant Data   

TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50107696(1,9-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)copy SMILEScopy InChI
Affinity DataKi:  0.776nMAssay Description:Displacement of [3H]NMS from human M4 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030223(CHEMBL3354068)copy SMILEScopy InChI
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H]NMS from human M3 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030223(CHEMBL3354068)copy SMILEScopy InChI
Affinity DataKi:  0.891nMAssay Description:Displacement of [3H]NMS from human M4 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030223(CHEMBL3354068)copy SMILEScopy InChI
Affinity DataKi:  0.912nMAssay Description:Displacement of [3H]NMS from human M1 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030224(CHEMBL3354069)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H]NMS from human M1 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030224(CHEMBL3354069)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]NMS from human M4 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030224(CHEMBL3354069)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]NMS from human M3 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030223(CHEMBL3354068)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]NMS from human M2 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030224(CHEMBL3354069)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]NMS from human M2 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50107696(1,9-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]NMS from human M1 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030223(CHEMBL3354068)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]NMS from human M5 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50107696(1,9-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)copy SMILEScopy InChI
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]NMS from human M3 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030224(CHEMBL3354069)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of [3H]NMS from human M5 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50107696(1,9-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]NMS from human M2 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50107696(1,9-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of [3H]NMS from human M5 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030222(CHEMBL3354067)copy SMILEScopy InChI
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]NMS from human M3 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030222(CHEMBL3354067)copy SMILEScopy InChI
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]NMS from human M5 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030225(CHEMBL3354070)copy SMILEScopy InChI
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]NMS from human M4 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030222(CHEMBL3354067)copy SMILEScopy InChI
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]NMS from human M1 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)copy SMILEScopy InChI
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]NMS from human M3 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030222(CHEMBL3354067)copy SMILEScopy InChI
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]NMS from human M4 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)copy SMILEScopy InChI
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]NMS from human M1 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)copy SMILEScopy InChI
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]NMS from human M2 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030225(CHEMBL3354070)copy SMILEScopy InChI
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]NMS from human M5 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)copy SMILEScopy InChI
Affinity DataKi:  9.30nMAssay Description:Displacement of [3H]NMS from human M5 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030225(CHEMBL3354070)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Displacement of [3H]NMS from human M3 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]NMS from human M4 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030222(CHEMBL3354067)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]NMS from human M2 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030225(CHEMBL3354070)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]NMS from human M1 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030242(CHEMBL3354071)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Displacement of [3H]NMS from human M4 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030221(CHEMBL3354066)copy SMILEScopy InChI
Affinity DataKi:  26nMAssay Description:Displacement of [3H]NMS from human M4 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030251(CHEMBL3354078)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Displacement of [3H]NMS from human M1 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030242(CHEMBL3354071)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Displacement of [3H]NMS from human M5 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030251(CHEMBL3354078)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:Displacement of [3H]NMS from human M4 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030242(CHEMBL3354071)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Displacement of [3H]NMS from human M1 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030242(CHEMBL3354071)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Displacement of [3H]NMS from human M3 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030251(CHEMBL3354078)copy SMILEScopy InChI
Affinity DataKi:  49nMAssay Description:Displacement of [3H]NMS from human M5 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030251(CHEMBL3354078)copy SMILEScopy InChI
Affinity DataKi:  58nMAssay Description:Displacement of [3H]NMS from human M3 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030221(CHEMBL3354066)copy SMILEScopy InChI
Affinity DataKi:  66nMAssay Description:Displacement of [3H]NMS from human M2 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030221(CHEMBL3354066)copy SMILEScopy InChI
Affinity DataKi:  78nMAssay Description:Displacement of [3H]NMS from human M1 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030251(CHEMBL3354078)copy SMILEScopy InChI
Affinity DataKi:  79nMAssay Description:Displacement of [3H]NMS from human M2 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030242(CHEMBL3354071)copy SMILEScopy InChI
Affinity DataKi:  85nMAssay Description:Displacement of [3H]NMS from human M2 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030225(CHEMBL3354070)copy SMILEScopy InChI
Affinity DataKi:  89nMAssay Description:Displacement of [3H]NMS from human M2 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030221(CHEMBL3354066)copy SMILEScopy InChI
Affinity DataKi:  93nMAssay Description:Displacement of [3H]NMS from human M3 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030249(CHEMBL3354077)copy SMILEScopy InChI
Affinity DataKi:  95nMAssay Description:Displacement of [3H]NMS from human M4 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030221(CHEMBL3354066)copy SMILEScopy InChI
Affinity DataKi:  102nMAssay Description:Displacement of [3H]NMS from human M5 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030248(CHEMBL3354076)copy SMILEScopy InChI
Affinity DataKi:  112nMAssay Description:Displacement of [3H]NMS from human M4 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030248(CHEMBL3354076)copy SMILEScopy InChI
Affinity DataKi:  123nMAssay Description:Displacement of [3H]NMS from human M1 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030247(CHEMBL3354075)copy SMILEScopy InChI
Affinity DataKi:  155nMAssay Description:Displacement of [3H]NMS from human M4 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50030249(CHEMBL3354077)copy SMILEScopy InChI
Affinity DataKi:  186nMAssay Description:Displacement of [3H]NMS from human M1 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NNBPubMed
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