Compile Data Set for Download or QSAR

Found 6 hits of Enzyme Inhibition Constant Data   

TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))copy SMILEScopy InChI
Affinity DataIC50: 150nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4HHDPubMed
TargetDeath-associated protein kinase 1(Homo sapiens (Human))
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))copy SMILEScopy InChI
Affinity DataIC50: 247nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4HHDPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4HHDPubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4HHDPubMed
TargetSerine/threonine-protein kinase PAK 5(Homo sapiens (Human))
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))copy SMILEScopy InChI
Affinity DataIC50: 5.60E+3nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4HHDPubMed
TargetDeath-associated protein kinase 1(Homo sapiens (Human))
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))copy SMILEScopy InChI
Affinity DataKd:  240nMpH: 7.5Assay Description:40 µL of a solution containing 350-500 µM of CPR005231 (compound 6) were titrated into the 200 µL sample cell containing 25-55 µM DAPK1 (AA 1-285) or...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4HHDPubMed
* indicates data uncertainty>20%