Compile Data Set for Download or QSAR

Found 37 hits of Enzyme Inhibition Constant Data   

TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102904(CHEMBL3394091)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102908(CHEMBL3393071)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102872(CHEMBL3394083)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50101585(CHEMBL3393986)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102878(CHEMBL3394082)copy SMILEScopy InChI
Affinity DataKi:  70nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102909(CHEMBL3394077)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102875(CHEMBL3394078)copy SMILEScopy InChI
Affinity DataKi:  110nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102906(CHEMBL3394089)copy SMILEScopy InChI
Affinity DataKi:  110nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102907(CHEMBL3394088)copy SMILEScopy InChI
Affinity DataKi:  120nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102903(CHEMBL3394092)copy SMILEScopy InChI
Affinity DataKi:  120nMAssay Description:Inhibition of human recombinant Abl kinase using [gamma-32P]ATP as substrate by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102908(CHEMBL3393071)copy SMILEScopy InChI
Affinity DataKi:  120nMAssay Description:Inhibition of human recombinant Abl kinase using [gamma-32P]ATP as substrate by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50101585(CHEMBL3393986)copy SMILEScopy InChI
Affinity DataKi:  130nMAssay Description:Inhibition of human recombinant Abl kinase using [gamma-32P]ATP as substrate by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102903(CHEMBL3394092)copy SMILEScopy InChI
Affinity DataKi:  130nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102871(CHEMBL3394084)copy SMILEScopy InChI
Affinity DataKi:  130nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102872(CHEMBL3394083)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Inhibition of human recombinant Abl kinase using [gamma-32P]ATP as substrate by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102904(CHEMBL3394091)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Inhibition of human recombinant Abl kinase using [gamma-32P]ATP as substrate by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50343430(CHEMBL1775036 | N-(3-Chlorophenyl)-1-(2-chloro-2-p...)copy SMILEScopy InChI
Affinity DataKi:  180nMAssay Description:Inhibition of human recombinant Abl kinase using [gamma-32P]ATP as substrate by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102887(CHEMBL3393983)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102877(CHEMBL3393979)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50343431(1-(2-Chloro-2-phenylethyl)-6-[(2-morpholin-4-yleth...)copy SMILEScopy InChI
Affinity DataKi:  210nMAssay Description:Inhibition of c-src kinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50343431(1-(2-Chloro-2-phenylethyl)-6-[(2-morpholin-4-yleth...)copy SMILEScopy InChI
Affinity DataKi:  220nMAssay Description:Inhibition of human recombinant Abl kinase using [gamma-32P]ATP as substrate by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102876(CHEMBL3393980)copy SMILEScopy InChI
Affinity DataKi:  230nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50343431(1-(2-Chloro-2-phenylethyl)-6-[(2-morpholin-4-yleth...)copy SMILEScopy InChI
Affinity DataKi:  240nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102869(CHEMBL3394086)copy SMILEScopy InChI
Affinity DataKi:  260nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50343430(CHEMBL1775036 | N-(3-Chlorophenyl)-1-(2-chloro-2-p...)copy SMILEScopy InChI
Affinity DataKi:  290nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102870(CHEMBL3394085)copy SMILEScopy InChI
Affinity DataKi:  300nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102878(CHEMBL3394082)copy SMILEScopy InChI
Affinity DataKi:  430nMAssay Description:Inhibition of human recombinant Abl kinase using [gamma-32P]ATP as substrate by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102910(CHEMBL3394076)copy SMILEScopy InChI
Affinity DataKi:  550nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102879(CHEMBL3393984)copy SMILEScopy InChI
Affinity DataKi:  620nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102874(CHEMBL3394087)copy SMILEScopy InChI
Affinity DataKi:  620nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102905(CHEMBL3394075)copy SMILEScopy InChI
Affinity DataKi:  790nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102881(CHEMBL3394081)copy SMILEScopy InChI
Affinity DataKi:  970nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102899(CHEMBL3393982)copy SMILEScopy InChI
Affinity DataKi:  1.06E+3nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102873(CHEMBL3393985)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102900(CHEMBL3394079)copy SMILEScopy InChI
Affinity DataKi:  1.44E+3nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102901(CHEMBL3393981)copy SMILEScopy InChI
Affinity DataKi:  1.46E+3nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena Via Aldo Moro 2

Curated by ChEMBL
LigandPNGBDBM50102889(CHEMBL3394080)copy SMILEScopy InChI
Affinity DataKi:  2.34E+3nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416ZTTPubMed
* indicates data uncertainty>20%