Compile Data Set for Download or QSAR

Found 24 hits of Enzyme Inhibition Constant Data   

TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043016(CHEMBL3355026 | US9718825, Example 3)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043018(CHEMBL3355028 | US9718825, Example 63)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043015(CHEMBL3355025 | US9718825, Example 1)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043021(CHEMBL3355031 | US9718825, Example 140)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043017(CHEMBL3355027)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043025(CHEMBL3355035 | US9718825, Example 520)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043019(CHEMBL3355029)copy SMILES
Affinity DataIC50: 1.5nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043020(CHEMBL3355030)copy SMILES
Affinity DataIC50: 1.5nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043023(CHEMBL3355033 | US9718825, Example 308)copy SMILES
Affinity DataIC50: 6.20nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043022(CHEMBL3355032)copy SMILEScopy InChI
Affinity DataIC50: 6.5nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043023(CHEMBL3355033 | US9718825, Example 308)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043026(CHEMBL3355036)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043021(CHEMBL3355031 | US9718825, Example 140)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043025(CHEMBL3355035 | US9718825, Example 520)copy SMILEScopy InChI
Affinity DataIC50: 61nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043017(CHEMBL3355027)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043019(CHEMBL3355029)copy SMILES
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043024(CHEMBL3355034 | US9718825, Example 310)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043022(CHEMBL3355032)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043020(CHEMBL3355030)copy SMILES
Affinity DataIC50: 170nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043024(CHEMBL3355034 | US9718825, Example 310)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043018(CHEMBL3355028 | US9718825, Example 63)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043026(CHEMBL3355036)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043016(CHEMBL3355026 | US9718825, Example 3)copy SMILEScopy InChI
Affinity DataIC50: 670nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC

Curated by ChEMBL
LigandPNGBDBM50043015(CHEMBL3355025 | US9718825, Example 1)copy SMILEScopy InChI
Affinity DataIC50: 830nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
* indicates data uncertainty>20%