Found 24 hits of Enzyme Inhibition Constant Data
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 6.20nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 61nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 390nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 830nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair