Found 65 hits of Enzyme Inhibition Constant Data
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of FGFR1 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Inhibition of FGFR2 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of FGFR4 (unknown origin)More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of FGFR3 (unknown origin)More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of FGFR1 (unknown origin)More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of FGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of FGFR3 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of FGFR2 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Inhibition of FGFR3 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 82nMAssay Description:Inhibition of FGFR1 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of FGFR1 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of FGFR4 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of FGFR2 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inhibition of FGFR3 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Inhibition of FGFR4 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of FGFR1 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of FGFR1 (unknown origin)More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of FGFR4 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 3.17E+3nMAssay Description:Inhibition of FGFR1 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 4.84E+3nMAssay Description:Inhibition of FGFR1 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 5.33E+3nMAssay Description:Inhibition of FGFR1 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 6.14E+3nMAssay Description:Inhibition of FGFR2 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 6.28E+3nMAssay Description:Inhibition of FGFR2 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 7.62E+3nMAssay Description:Inhibition of FGFR2 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 8.39E+3nMAssay Description:Inhibition of FGFR2 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 9.13E+3nMAssay Description:Inhibition of FGFR2 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 9.13E+3nMAssay Description:Inhibition of FGFR1 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 9.13E+3nMAssay Description:Inhibition of FGFR2 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 9.58E+3nMAssay Description:Inhibition of FGFR2 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 9.59E+3nMAssay Description:Inhibition of FGFR1 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of FGFR1 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of FGFR1 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of FGFR2 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of FGFR2 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of FGFR1 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.52E+4nMAssay Description:Inhibition of FGFR1 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.52E+4nMAssay Description:Inhibition of FGFR1 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.57E+4nMAssay Description:Inhibition of FGFR2 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of FGFR2 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.77E+4nMAssay Description:Inhibition of FGFR2 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.78E+4nMAssay Description:Inhibition of FGFR1 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of FGFR3 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.96E+4nMAssay Description:Inhibition of FGFR3 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.96E+4nMAssay Description:Inhibition of FGFR3 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.98E+4nMAssay Description:Inhibition of FGFR3 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of FGFR4 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of FGFR4 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of FGFR4 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of FGFR3 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Health Science Center Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of FGFR4 (unknown origin) after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
![](/img/powered_by_small.gif)