Compile Data Set for Download or QSAR

Found 143 hits of Enzyme Inhibition Constant Data   

TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105928(CHEMBL3598047)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106011(CHEMBL3598077)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105992(CHEMBL3598061)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105981(CHEMBL3598052)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105930(CHEMBL3598049)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105982(CHEMBL3598053)copy SMILEScopy InChI
Affinity DataIC50: 4.80nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105985(CHEMBL3598055)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105988(CHEMBL3598056)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105933(CHEMBL3598051)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105990(CHEMBL3598057)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106002(CHEMBL3598070)copy SMILEScopy InChI
Affinity DataIC50: 5.10nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106003(CHEMBL3598071)copy SMILEScopy InChI
Affinity DataIC50: 5.20nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105995(CHEMBL3598063)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106009(CHEMBL3598076)copy SMILEScopy InChI
Affinity DataIC50: 6.20nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106007(CHEMBL3598074)copy SMILEScopy InChI
Affinity DataIC50: 6.40nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106008(CHEMBL3598075)copy SMILEScopy InChI
Affinity DataIC50: 8.40nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105929(CHEMBL3598048)copy SMILEScopy InChI
Affinity DataIC50: 8.60nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105984(CHEMBL3598054)copy SMILEScopy InChI
Affinity DataIC50: 9.20nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105998(CHEMBL3598065)copy SMILEScopy InChI
Affinity DataIC50: 9.40nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105991(CHEMBL3598060)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105932(CHEMBL3598050)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106004(CHEMBL3598072)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105997(CHEMBL3598064)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106000(CHEMBL3598066)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105925(CHEMBL3598044)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106001(CHEMBL3598068)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105924(CHEMBL3598043)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105919(CHEMBL3596632)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105922(CHEMBL3598041)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106005(CHEMBL3598073)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105927(CHEMBL3598046)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105993(CHEMBL3598062)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105926(CHEMBL3598045)copy SMILEScopy InChI
Affinity DataIC50: 76nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105920(CHEMBL3598040)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105921(CHEMBL3596216)copy SMILEScopy InChI
Affinity DataIC50: 530nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105923(CHEMBL3598042)copy SMILEScopy InChI
Affinity DataIC50: 610nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106013(CHEMBL3598079)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+3nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106012(CHEMBL3598078)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105919(CHEMBL3596632)copy SMILEScopy InChI
Affinity DataEC50:  98nMAssay Description:Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106121(CHEMBL3598059)copy SMILEScopy InChI
Affinity DataEC50:  15nMAssay Description:Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106000(CHEMBL3598066)copy SMILEScopy InChI
Affinity DataEC50:  37nMAssay Description:Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106008(CHEMBL3598075)copy SMILEScopy InChI
Affinity DataEC50:  17nMAssay Description:Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106009(CHEMBL3598076)copy SMILEScopy InChI
Affinity DataEC50:  13nMAssay Description:Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Mus musculus)
Biogen

Curated by ChEMBL
LigandPNGBDBM50105925(CHEMBL3598044)copy SMILEScopy InChI
Affinity DataEC50:  3.11E+3nMAssay Description:Inverse agonist activity at RORgamma in C57BL/6 mouse splenocytes assessed as reduction of IL-17 production after 2 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Mus musculus)
Biogen

Curated by ChEMBL
LigandPNGBDBM50105928(CHEMBL3598047)copy SMILEScopy InChI
Affinity DataEC50:  38nMAssay Description:Inverse agonist activity at RORgamma in C57BL/6 mouse splenocytes assessed as reduction of IL-17 production after 2 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-gamma(Mus musculus)
Biogen

Curated by ChEMBL
LigandPNGBDBM50105991(CHEMBL3598060)copy SMILEScopy InChI
Affinity DataEC50:  134nMAssay Description:Inverse agonist activity at RORgamma in C57BL/6 mouse splenocytes assessed as reduction of IL-17 production after 2 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-alpha(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105925(CHEMBL3598044)copy SMILEScopy InChI
Affinity DataEC50:  1.20E+3nMAssay Description:Inverse agonist activity at RORalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-alpha(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105982(CHEMBL3598053)copy SMILEScopy InChI
Affinity DataEC50:  2.00E+3nMAssay Description:Inverse agonist activity at RORalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-alpha(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106011(CHEMBL3598077)copy SMILEScopy InChI
Affinity DataEC50:  2.20E+3nMAssay Description:Inverse agonist activity at RORalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105932(CHEMBL3598050)copy SMILEScopy InChI
Affinity DataEC50:  1.10E+3nMAssay Description:Inverse agonist activity at RORbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X3508HPubMed
Displayed 1 to 50 (of 143 total ) | Next | Last >>* indicates data uncertainty>20%