Compile Data Set for Download or QSAR

Found 72 hits of Enzyme Inhibition Constant Data   

TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50072394(1-[3-(1H-4-imidazolyl)-2-(5-oxotetrahydro-1H-2-pyr...)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50072394(1-[3-(1H-4-imidazolyl)-2-(5-oxotetrahydro-1H-2-pyr...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109025(CHEMBL3600444)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109027(CHEMBL3600446)copy SMILES
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109028(CHEMBL3600447)copy SMILES
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109039(CHEMBL3600454)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109018(CHEMBL3601784)copy SMILES
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109022(CHEMBL3601785)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109023(CHEMBL3601786)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109026(CHEMBL3600445)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109035(CHEMBL3600450)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109040(CHEMBL3601782)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109038(CHEMBL3600453)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109033(CHEMBL3600448)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109027(CHEMBL3600446)copy SMILES
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109017(CHEMBL3601783)copy SMILES
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109037(CHEMBL3600452)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109041(CHEMBL3601781)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109036(CHEMBL3600451)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109035(CHEMBL3600450)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109025(CHEMBL3600444)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109028(CHEMBL3600447)copy SMILES
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109033(CHEMBL3600448)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109034(CHEMBL3600449)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109039(CHEMBL3600454)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109034(CHEMBL3600449)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109026(CHEMBL3600445)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109023(CHEMBL3601786)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109022(CHEMBL3601785)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109037(CHEMBL3600452)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109036(CHEMBL3600451)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109041(CHEMBL3601781)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109038(CHEMBL3600453)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109018(CHEMBL3601784)copy SMILES
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109017(CHEMBL3601783)copy SMILES
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109040(CHEMBL3601782)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109017(CHEMBL3601783)copy SMILES
Affinity DataEC50:  290nMAssay Description:Agonist activity at mouse TRH-R2 expressed in HEK293 cells assessed as induction of changes in intracellular Ca2+ level by FLIPR methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50072394(1-[3-(1H-4-imidazolyl)-2-(5-oxotetrahydro-1H-2-pyr...)copy SMILEScopy InChI
Affinity DataEC50:  1nMAssay Description:Agonist activity at mouse TRH-R1 expressed in HEK293 cells assessed as induction of changes in intracellular Ca2+ level by FLIPR methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109035(CHEMBL3600450)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at mouse TRH-R1 expressed in HEK293 cells assessed as induction of changes in intracellular Ca2+ level by FLIPR methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109039(CHEMBL3600454)copy SMILEScopy InChI
Affinity DataEC50:  100nMAssay Description:Agonist activity at mouse TRH-R2 expressed in HEK293 cells assessed as induction of changes in intracellular Ca2+ level by FLIPR methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109018(CHEMBL3601784)copy SMILES
Affinity DataEC50:  310nMAssay Description:Agonist activity at mouse TRH-R2 expressed in HEK293 cells assessed as induction of changes in intracellular Ca2+ level by FLIPR methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109034(CHEMBL3600449)copy SMILEScopy InChI
Affinity DataEC50:  4nMAssay Description:Agonist activity at mouse TRH-R2 expressed in HEK293 cells assessed as induction of changes in intracellular Ca2+ level by FLIPR methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50072394(1-[3-(1H-4-imidazolyl)-2-(5-oxotetrahydro-1H-2-pyr...)copy SMILEScopy InChI
Affinity DataEC50:  0.520nMAssay Description:Agonist activity at mouse TRH-R2 expressed in HEK293 cells assessed as induction of changes in intracellular Ca2+ level by FLIPR methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109018(CHEMBL3601784)copy SMILES
Affinity DataEC50:  1.13E+4nMAssay Description:Agonist activity at mouse TRH-R1 expressed in HEK293 cells assessed as induction of changes in intracellular Ca2+ level by FLIPR methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109036(CHEMBL3600451)copy SMILEScopy InChI
Affinity DataEC50:  530nMAssay Description:Agonist activity at mouse TRH-R2 expressed in HEK293 cells assessed as induction of changes in intracellular Ca2+ level by FLIPR methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109025(CHEMBL3600444)copy SMILEScopy InChI
Affinity DataEC50:  50nMAssay Description:Agonist activity at mouse TRH-R2 expressed in HEK293 cells assessed as induction of changes in intracellular Ca2+ level by FLIPR methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109038(CHEMBL3600453)copy SMILEScopy InChI
Affinity DataEC50:  2.54E+3nMAssay Description:Agonist activity at mouse TRH-R1 expressed in HEK293 cells assessed as induction of changes in intracellular Ca2+ level by FLIPR methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109017(CHEMBL3601783)copy SMILES
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity at mouse TRH-R1 expressed in HEK293 cells assessed as induction of changes in intracellular Ca2+ level by FLIPR methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109023(CHEMBL3601786)copy SMILEScopy InChI
Affinity DataEC50:  7.21E+3nMAssay Description:Agonist activity at mouse TRH-R1 expressed in HEK293 cells assessed as induction of changes in intracellular Ca2+ level by FLIPR methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
TargetThyrotropin-releasing hormone receptor(Mus musculus)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50109022(CHEMBL3601785)copy SMILEScopy InChI
Affinity DataEC50:  30nMAssay Description:Agonist activity at mouse TRH-R2 expressed in HEK293 cells assessed as induction of changes in intracellular Ca2+ level by FLIPR methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NZ9PubMed
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