Compile Data Set for Download or QSAR

Found 50 hits of Enzyme Inhibition Constant Data   

TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111480(CHEMBL3604943)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM149404(AVL-301 | CHEMBL3545308 | CNX-419 | CO-1686 | Roci...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50383274(CHEMBL1229592 | US10167264, WZ4002 | US9670213, WZ...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111473(CHEMBL3604937)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of cSrc T338M/S345C mutant (unknown origin) pre-incubated for 30 mins before substrate and ATP addition by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111472(CHEMBL3604921)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of cSrc T338M/S345C mutant (unknown origin) pre-incubated for 30 mins before substrate and ATP addition by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111470(CHEMBL1232944)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibition of cSrc T338M/S345C mutant (unknown origin) pre-incubated for 30 mins before substrate and ATP addition by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111471(CHEMBL3604910)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of cSrc T338M/S345C mutant (unknown origin) pre-incubated for 30 mins before substrate and ATP addition by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111471(CHEMBL3604910)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of cSrc T338M mutant (unknown origin) pre-incubated for 30 mins before substrate and ATP addition by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111470(CHEMBL1232944)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:Inhibition of cSrc T338M mutant (unknown origin) pre-incubated for 30 mins before substrate and ATP addition by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111472(CHEMBL3604921)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of cSrc T338M mutant (unknown origin) pre-incubated for 30 mins before substrate and ATP addition by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111470(CHEMBL1232944)copy SMILEScopy InChI
Affinity DataIC50: 211nMAssay Description:Inhibition of wild type cSrc (251 to 533 residues) (unknown origin) pre-incubated for 30 mins before substrate and ATP addition by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM153729(N-(3-((4-((5-Methyl-1H-pyrazol-3-yl)amino)-6-(4-me...)copy SMILEScopy InChI
Affinity DataIC50: 254nMAssay Description:Inhibition of cSrc T338M mutant (unknown origin) pre-incubated for 30 mins before substrate and ATP addition by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111474(CHEMBL3604938)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of cSrc T338M/S345C mutant (unknown origin) pre-incubated for 30 mins before substrate and ATP addition by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111471(CHEMBL3604910)copy SMILEScopy InChI
Affinity DataIC50: 336nMAssay Description:Inhibition of wild type cSrc (251 to 533 residues) (unknown origin) pre-incubated for 30 mins before substrate and ATP addition by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM153729(N-(3-((4-((5-Methyl-1H-pyrazol-3-yl)amino)-6-(4-me...)copy SMILEScopy InChI
Affinity DataIC50: 349nMAssay Description:Inhibition of cSrc T338M/S345C mutant (unknown origin) pre-incubated for 30 mins before substrate and ATP addition by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111482(CHEMBL3604917)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111484(CHEMBL3604920)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111490(CHEMBL3604912)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111450(CHEMBL3604935)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111473(CHEMBL3604937)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111475(CHEMBL3604936)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111478(CHEMBL3604940)copy SMILEScopy InChI
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111485(CHEMBL3604922)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111479(CHEMBL3604941)copy SMILEScopy InChI
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111487(CHEMBL3604915)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM153717(N-(5-Methyl-1H-pyrazol-3-yl)-6-(4-methylpiperazin-...)copy SMILEScopy InChI
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111477(CHEMBL3604939)copy SMILEScopy InChI
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111447(CHEMBL3604933)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM153730(N-(4-((4-((5-Methyl-1H-pyrazol-3-yl)amino)-6-(4-me...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111474(CHEMBL3604938)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111493(CHEMBL3604919)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111489(CHEMBL3604913)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111491(CHEMBL3604911)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111470(CHEMBL1232944)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM153718(N-(5-Methyl-1H-pyrazol-3-yl)-6-(4-methylpiperazin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111472(CHEMBL3604921)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM153728(2-(4-Aminophenoxy)-N-(5-methyl-1H-pyrazol-3-yl)-6-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111481(CHEMBL3604916)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111488(CHEMBL3604914)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111442(CHEMBL3604932)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111436(CHEMBL3604931)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111397(CHEMBL3604929)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM153716(N-(5-Methyl-1H-pyrazol-3-yl)-6-(4-methylpiperazin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111492(CHEMBL3604942)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111483(CHEMBL3604918)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM153729(N-(3-((4-((5-Methyl-1H-pyrazol-3-yl)amino)-6-(4-me...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111486(CHEMBL3604923)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111471(CHEMBL3604910)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50111449(CHEMBL3604934)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type EGFR (unknown origin) expressed in Sf9 cells pre-incubated for 30 mins before substrate and ATP addition by homogeneous time-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1G59PubMed
* indicates data uncertainty>20%