Compile Data Set for Download or QSAR

Found 7 hits of Enzyme Inhibition Constant Data   

TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Ume£ University

Curated by ChEMBL
LigandPNGBDBM50500150(CHEMBL3746821)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at PPARgamma (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W95D6BPubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Ume£ University

Curated by ChEMBL
LigandPNGBDBM50500150(CHEMBL3746821)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at RXRalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W95D6BPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Ume£ University

Curated by ChEMBL
LigandPNGBDBM50500150(CHEMBL3746821)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at PPARalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W95D6BPubMed
TargetBile acid receptor(Homo sapiens (Human))
Ume£ University

Curated by ChEMBL
LigandPNGBDBM50500150(CHEMBL3746821)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at FXR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W95D6BPubMed
TargetLipoprotein lipase(Bos taurus)
Ume£ University

Curated by ChEMBL
LigandPNGBDBM50500148(CHEMBL3746381)copy SMILEScopy InChI
Affinity DataEC50:  6.60E+3nMAssay Description:Induction of bovine LPL stabilization using intralipid as substrate preincubated for 10 mins with human recombinant ANGPTL4 followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W95D6BPubMed
TargetLipoprotein lipase(Bos taurus)
Ume£ University

Curated by ChEMBL
LigandPNGBDBM50500149(CHEMBL3747367)copy SMILEScopy InChI
Affinity DataEC50:  5.00E+3nMAssay Description:Induction of bovine LPL stabilization using intralipid as substrate preincubated for 10 mins with human recombinant ANGPTL4 followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W95D6BPubMed
TargetLipoprotein lipase(Bos taurus)
Ume£ University

Curated by ChEMBL
LigandPNGBDBM50500150(CHEMBL3746821)copy SMILEScopy InChI
Affinity DataEC50:  6.00E+3nMAssay Description:Induction of bovine LPL stabilization using intralipid as substrate preincubated for 10 mins with human recombinant ANGPTL4 followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W95D6BPubMed
* indicates data uncertainty>20%