Found 23 hits of Enzyme Inhibition Constant Data
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.160nMAssay Description:Inhibition of GST-tagged TNKS2 (873 to 1166 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.170nMAssay Description:Inhibition of GST-tagged TNKS2 (873 to 1166 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.180nMAssay Description:Inhibition of GST-tagged TNKS1 (1023 to 1327 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.180nMAssay Description:Inhibition of GST-tagged TNKS2 (873 to 1166 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.190nMAssay Description:Inhibition of GST-tagged TNKS2 (873 to 1166 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of GST-tagged TNKS1 (1023 to 1327 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.240nMAssay Description:Inhibition of GST-tagged TNKS1 (1023 to 1327 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.280nMAssay Description:Inhibition of GST-tagged TNKS2 (873 to 1166 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of GST-tagged TNKS1 (1023 to 1327 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.810nMAssay Description:Inhibition of GST-tagged TNKS1 (1023 to 1327 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 3.90nMAssay Description:Inhibition of GST-tagged TNKS2 (873 to 1166 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 8.5nMAssay Description:Inhibition of GST-tagged TNKS1 (1023 to 1327 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human recombinant His-tagged PARP1 autoparsylation expressed in sf21 cells using NAD and biotinylated NAD incubated for 150 mins by HTR...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 730nMAssay Description:Inhibition of human recombinant His-tagged PARP1 autoparsylation expressed in sf21 cells using NAD and biotinylated NAD incubated for 150 mins by HTR...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant His-tagged PARP1 autoparsylation expressed in sf21 cells using NAD and biotinylated NAD incubated for 150 mins by HTR...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human recombinant His-tagged PARP1 autoparsylation expressed in sf21 cells using NAD and biotinylated NAD incubated for 150 mins by HTR...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human recombinant His-tagged PARP1 autoparsylation expressed in sf21 cells using NAD and biotinylated NAD incubated for 150 mins by HTR...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1/tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataEC50: 0.260nMAssay Description:Inhibition of tankyrase in human DLD1 cells assessed as increase in axin2 level after 24 hrs by fluorescence analysisMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1/tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataEC50: 2.90nMAssay Description:Inhibition of tankyrase in human DLD1 cells assessed as increase in axin2 level after 24 hrs by fluorescence analysisMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1/tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataEC50: 48nMAssay Description:Inhibition of tankyrase in human DLD1 cells assessed as increase in axin2 level after 24 hrs by fluorescence analysisMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1/tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataEC50: 21nMAssay Description:Inhibition of tankyrase in human DLD1 cells assessed as increase in axin2 level after 24 hrs by fluorescence analysisMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1/tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataEC50: 0.220nMAssay Description:Inhibition of tankyrase in human DLD1 cells assessed as increase in axin2 level after 24 hrs by fluorescence analysisMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1/tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataEC50: 1.30nMAssay Description:Inhibition of tankyrase in human DLD1 cells assessed as increase in axin2 level after 24 hrs by fluorescence analysisMore data for this Ligand-Target Pair
