Compile Data Set for Download or QSAR

Found 183 hits of Enzyme Inhibition Constant Data   

TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187587(CHEMBL3827598)copy SMILEScopy InChI
Affinity DataKi:  56nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187585(CHEMBL3827074)copy SMILEScopy InChI
Affinity DataKi:  72nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187591(CHEMBL3827331)copy SMILEScopy InChI
Affinity DataKi:  80nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187591(CHEMBL3827331)copy SMILEScopy InChI
Affinity DataKi:  109nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187588(CHEMBL3827201)copy SMILEScopy InChI
Affinity DataKi:  127nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187660(CHEMBL3828002)copy SMILEScopy InChI
Affinity DataKi:  131nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187584(CHEMBL3827187)copy SMILEScopy InChI
Affinity DataKi:  137nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187664(CHEMBL3828555)copy SMILEScopy InChI
Affinity DataKi:  172nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187592(CHEMBL3827301)copy SMILEScopy InChI
Affinity DataKi:  174nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187586(CHEMBL3827623)copy SMILEScopy InChI
Affinity DataKi:  175nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187662(CHEMBL3827267)copy SMILEScopy InChI
Affinity DataKi:  180nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187660(CHEMBL3828002)copy SMILEScopy InChI
Affinity DataKi:  184nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187605(CHEMBL3827298)copy SMILEScopy InChI
Affinity DataKi:  254nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187593(CHEMBL3827922)copy SMILEScopy InChI
Affinity DataKi:  268nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187590(CHEMBL3827583)copy SMILEScopy InChI
Affinity DataKi:  271nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187659(CHEMBL3827716)copy SMILEScopy InChI
Affinity DataKi:  297nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187591(CHEMBL3827331)copy SMILEScopy InChI
Affinity DataKi:  310nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A3 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187664(CHEMBL3828555)copy SMILEScopy InChI
Affinity DataKi:  337nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187676(CHEMBL3828401)copy SMILEScopy InChI
Affinity DataKi:  338nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187589(CHEMBL3827859)copy SMILEScopy InChI
Affinity DataKi:  339nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187676(CHEMBL3828401)copy SMILEScopy InChI
Affinity DataKi:  347nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187674(CHEMBL3828658)copy SMILEScopy InChI
Affinity DataKi:  370nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187674(CHEMBL3828658)copy SMILEScopy InChI
Affinity DataKi:  464nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187655(CHEMBL3827920)copy SMILEScopy InChI
Affinity DataKi: >500nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187661(CHEMBL3828044)copy SMILEScopy InChI
Affinity DataKi: >500nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187590(CHEMBL3827583)copy SMILEScopy InChI
Affinity DataKi: >500nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187660(CHEMBL3828002)copy SMILEScopy InChI
Affinity DataKi:  518nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187587(CHEMBL3827598)copy SMILEScopy InChI
Affinity DataKi:  539nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine receptor A1 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187591(CHEMBL3827331)copy SMILEScopy InChI
Affinity DataKi:  546nMAssay Description:Displacement of [3H]MSX2 from recombinant human adenosine receptor A2a expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187589(CHEMBL3827859)copy SMILEScopy InChI
Affinity DataKi:  559nMAssay Description:Displacement of [3H]MSX2 from recombinant human adenosine receptor A2a expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187591(CHEMBL3827331)copy SMILEScopy InChI
Affinity DataKi:  566nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187666(CHEMBL3827653)copy SMILEScopy InChI
Affinity DataKi:  567nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187596(CHEMBL3827016)copy SMILEScopy InChI
Affinity DataKi:  585nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187660(CHEMBL3828002)copy SMILEScopy InChI
Affinity DataKi:  619nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A3 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187676(CHEMBL3828401)copy SMILEScopy InChI
Affinity DataKi:  633nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A3 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187595(CHEMBL3828343)copy SMILEScopy InChI
Affinity DataKi:  645nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187599(CHEMBL3828237)copy SMILEScopy InChI
Affinity DataKi:  653nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187585(CHEMBL3827074)copy SMILEScopy InChI
Affinity DataKi:  658nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine receptor A1 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187676(CHEMBL3828401)copy SMILEScopy InChI
Affinity DataKi:  658nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187674(CHEMBL3828658)copy SMILEScopy InChI
Affinity DataKi:  663nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187585(CHEMBL3827074)copy SMILEScopy InChI
Affinity DataKi:  666nMAssay Description:Displacement of [3H]MSX2 from recombinant human adenosine receptor A2a expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187588(CHEMBL3827201)copy SMILEScopy InChI
Affinity DataKi:  713nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine receptor A1 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187592(CHEMBL3827301)copy SMILEScopy InChI
Affinity DataKi:  738nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187661(CHEMBL3828044)copy SMILEScopy InChI
Affinity DataKi:  785nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187655(CHEMBL3827920)copy SMILEScopy InChI
Affinity DataKi:  853nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187667(CHEMBL3827365)copy SMILEScopy InChI
Affinity DataKi:  859nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187664(CHEMBL3828555)copy SMILEScopy InChI
Affinity DataKi:  890nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A3 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187656(CHEMBL3093326)copy SMILEScopy InChI
Affinity DataKi:  893nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187588(CHEMBL3827201)copy SMILEScopy InChI
Affinity DataKi:  921nMAssay Description:Displacement of [3H]MSX2 from recombinant human adenosine receptor A2a expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187585(CHEMBL3827074)copy SMILEScopy InChI
Affinity DataKi:  989nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SQ5PubMed
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