Found 27 hits of Enzyme Inhibition Constant Data
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataKi: 800nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataKi: 2.50E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataKi: 4.70E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataKi: 6.00E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 3.08E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Fyn expressed in baculovirus infected Sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 4.32E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Fyn expressed in baculovirus infected Sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of Flt3 (unknown origin) using KVEKIGEGTYGVVYK as substrate after 10 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 5.71E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Fyn expressed in baculovirus infected Sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 5.82E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Fyn expressed in baculovirus infected Sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of Flt3 (unknown origin) using KVEKIGEGTYGVVYK as substrate after 10 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 6.10E+4nMAssay Description:Inhibition of Flt3 (unknown origin) using KVEKIGEGTYGVVYK as substrate after 10 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 6.10E+4nMAssay Description:Inhibition of Flt3 (unknown origin) using KVEKIGEGTYGVVYK as substrate after 10 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Fyn expressed in baculovirus infected Sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 6.40E+4nMAssay Description:Inhibition of Flt3 (unknown origin) using KVEKIGEGTYGVVYK as substrate after 10 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 6.80E+4nMAssay Description:Inhibition of Flt3 (unknown origin) using KVEKIGEGTYGVVYK as substrate after 10 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of Abl (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 7.04E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Fyn expressed in baculovirus infected Sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 7.20E+4nMAssay Description:Inhibition of Flt3 (unknown origin) using KVEKIGEGTYGVVYK as substrate after 10 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 7.60E+4nMAssay Description:Inhibition of Flt3 (unknown origin) using KVEKIGEGTYGVVYK as substrate after 10 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 7.60E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Fyn expressed in baculovirus infected Sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£ degli Studi di Genova
Curated by ChEMBL
Universit£ degli Studi di Genova
Curated by ChEMBL
Affinity DataIC50: 8.86E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Fyn expressed in baculovirus infected Sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
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