Compile Data Set for Download or QSAR

Found 27 hits of Enzyme Inhibition Constant Data   

TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230317(CHEMBL4091022)copy SMILEScopy InChI
Affinity DataKi:  500nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230313(CHEMBL4068876)copy SMILEScopy InChI
Affinity DataKi:  700nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230311(CHEMBL4063136)copy SMILEScopy InChI
Affinity DataKi:  800nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230318(CHEMBL4103914)copy SMILEScopy InChI
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230316(CHEMBL4088440)copy SMILEScopy InChI
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230321(CHEMBL4073713)copy SMILEScopy InChI
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230319(CHEMBL4060213)copy SMILEScopy InChI
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230320(CHEMBL4100526)copy SMILEScopy InChI
Affinity DataKi:  4.70E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230312(CHEMBL4098763)copy SMILEScopy InChI
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230315(CHEMBL4096164)copy SMILEScopy InChI
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230311(CHEMBL4063136)copy SMILEScopy InChI
Affinity DataIC50: 3.08E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Fyn expressed in baculovirus infected Sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230317(CHEMBL4091022)copy SMILEScopy InChI
Affinity DataIC50: 4.32E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Fyn expressed in baculovirus infected Sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230313(CHEMBL4068876)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of Flt3 (unknown origin) using KVEKIGEGTYGVVYK as substrate after 10 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230321(CHEMBL4073713)copy SMILEScopy InChI
Affinity DataIC50: 5.71E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Fyn expressed in baculovirus infected Sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230313(CHEMBL4068876)copy SMILEScopy InChI
Affinity DataIC50: 5.82E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Fyn expressed in baculovirus infected Sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230317(CHEMBL4091022)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of Flt3 (unknown origin) using KVEKIGEGTYGVVYK as substrate after 10 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230320(CHEMBL4100526)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+4nMAssay Description:Inhibition of Flt3 (unknown origin) using KVEKIGEGTYGVVYK as substrate after 10 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230321(CHEMBL4073713)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+4nMAssay Description:Inhibition of Flt3 (unknown origin) using KVEKIGEGTYGVVYK as substrate after 10 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230318(CHEMBL4103914)copy SMILEScopy InChI
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Fyn expressed in baculovirus infected Sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230316(CHEMBL4088440)copy SMILEScopy InChI
Affinity DataIC50: 6.40E+4nMAssay Description:Inhibition of Flt3 (unknown origin) using KVEKIGEGTYGVVYK as substrate after 10 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230315(CHEMBL4096164)copy SMILEScopy InChI
Affinity DataIC50: 6.80E+4nMAssay Description:Inhibition of Flt3 (unknown origin) using KVEKIGEGTYGVVYK as substrate after 10 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230317(CHEMBL4091022)copy SMILEScopy InChI
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of Abl (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230312(CHEMBL4098763)copy SMILEScopy InChI
Affinity DataIC50: 7.04E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Fyn expressed in baculovirus infected Sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230318(CHEMBL4103914)copy SMILEScopy InChI
Affinity DataIC50: 7.20E+4nMAssay Description:Inhibition of Flt3 (unknown origin) using KVEKIGEGTYGVVYK as substrate after 10 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230312(CHEMBL4098763)copy SMILEScopy InChI
Affinity DataIC50: 7.60E+4nMAssay Description:Inhibition of Flt3 (unknown origin) using KVEKIGEGTYGVVYK as substrate after 10 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230316(CHEMBL4088440)copy SMILEScopy InChI
Affinity DataIC50: 7.60E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Fyn expressed in baculovirus infected Sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£ degli Studi di Genova

Curated by ChEMBL
LigandPNGBDBM50230315(CHEMBL4096164)copy SMILEScopy InChI
Affinity DataIC50: 8.86E+4nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Fyn expressed in baculovirus infected Sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
* indicates data uncertainty>20%