Compile Data Set for Download or QSAR

Found 5 hits of Enzyme Inhibition Constant Data   

TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50334986(4,4-Difluoro-cyclohexanecarboxylic acid {(S)-3-[(1...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of CCR5 in human TZM-bl cells infected with HIV1 Bal R5 assessed as antiviral activity by measuring reduction in viral infection pre-incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GTWPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Peking University

Curated by ChEMBL
LigandPNGBDBM50453729(CHEMBL4206186)copy SMILEScopy InChI
Affinity DataKd:  1.15E+5nMAssay Description:Binding affinity to HIV1 integrase by surface plasma resonance methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GTWPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Peking University

Curated by ChEMBL
LigandPNGBDBM50453728(CHEMBL4218163)copy SMILEScopy InChI
Affinity DataKd:  1.60E+5nMAssay Description:Binding affinity to HIV1 integrase by surface plasma resonance methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GTWPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Peking University

Curated by ChEMBL
LigandPNGBDBM50453727(CHEMBL4214002)copy SMILEScopy InChI
Affinity DataKd:  2.07E+5nMAssay Description:Binding affinity to HIV1 integrase by surface plasma resonance methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GTWPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Peking University

Curated by ChEMBL
LigandPNGBDBM50453730(CHEMBL4206051)copy SMILEScopy InChI
Affinity DataKd:  1.42E+5nMAssay Description:Binding affinity to HIV1 integrase by surface plasma resonance methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GTWPubMed
* indicates data uncertainty>20%