Compile Data Set for Download or QSAR

Found 85 hits of Enzyme Inhibition Constant Data   

TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)copy SMILEScopy InChI
Affinity DataKi:  4.80nMAssay Description:Reversible inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245603(CHEMBL4096207)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Reversible inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245586(CHEMBL4077123)copy SMILEScopy InChI
Affinity DataKi:  8.90nMAssay Description:Reversible inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245587(CHEMBL4077064 | US10000483, Compound II-4)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Reversible inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50161162(AVL-292 | CC-292 | Spebrutinib | US10596172, Compo...)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Reversible inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50020471(CHEMBL3290142)copy SMILEScopy InChI
Affinity DataKi:  27nMAssay Description:Reversible inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245588(CHEMBL4085868)copy SMILEScopy InChI
Affinity DataKi:  113nMAssay Description:Reversible inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50403056(CHEMBL2216827 | US10596172, Compound I-342 | US108...)copy SMILEScopy InChI
Affinity DataKi:  209nMAssay Description:Reversible inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245588(CHEMBL4085868)copy SMILEScopy InChI
Affinity DataIC50: 5.80nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245586(CHEMBL4077123)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
TargetCytoplasmic tyrosine-protein kinase BMX(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged BMX expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50161162(AVL-292 | CC-292 | Spebrutinib | US10596172, Compo...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50403056(CHEMBL2216827 | US10596172, Compound I-342 | US108...)copy SMILEScopy InChI
Affinity DataIC50: 9.5nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245587(CHEMBL4077064 | US10000483, Compound II-4)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245603(CHEMBL4096207)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245613(CHEMBL4074840)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245635(CHEMBL4076543)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245602(CHEMBL4088999)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetCytoplasmic tyrosine-protein kinase BMX(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50020471(CHEMBL3290142)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged BMX expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50020471(CHEMBL3290142)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245642(CHEMBL4059850)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245614(CHEMBL4066223)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245612(CHEMBL4101519)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetCytoplasmic tyrosine-protein kinase BMX(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245587(CHEMBL4077064 | US10000483, Compound II-4)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged BMX expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245617(CHEMBL4067226)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245632(CHEMBL4077618)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245646(CHEMBL4066966)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245636(CHEMBL4071818)copy SMILEScopy InChI
Affinity DataIC50: 68nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50020471(CHEMBL3290142)copy SMILEScopy InChI
Affinity DataIC50: 72nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged wild-type EGFR (695 to end residues) expressed in baculovirus infected Sf9 insect cells using p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245628(CHEMBL4064326)copy SMILEScopy InChI
Affinity DataIC50: 76nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245627(CHEMBL4093610)copy SMILEScopy InChI
Affinity DataIC50: 86nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245639(CHEMBL4088485)copy SMILEScopy InChI
Affinity DataIC50: 89nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245630(CHEMBL4074645)copy SMILEScopy InChI
Affinity DataIC50: 114nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)copy SMILEScopy InChI
Affinity DataIC50: 123nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged wild-type EGFR (695 to end residues) expressed in baculovirus infected Sf9 insect cells using p...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245604(CHEMBL4076040)copy SMILEScopy InChI
Affinity DataIC50: 127nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)copy SMILEScopy InChI
Affinity DataIC50: 146nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245643(CHEMBL4081428)copy SMILEScopy InChI
Affinity DataIC50: 163nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245599(CHEMBL4105457)copy SMILEScopy InChI
Affinity DataIC50: 187nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245637(CHEMBL4093800)copy SMILEScopy InChI
Affinity DataIC50: 197nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245629(CHEMBL4081768)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245634(CHEMBL4063526)copy SMILEScopy InChI
Affinity DataIC50: 231nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245645(CHEMBL4103674)copy SMILEScopy InChI
Affinity DataIC50: 244nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245626(CHEMBL4094515)copy SMILEScopy InChI
Affinity DataIC50: 273nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245618(CHEMBL4071893)copy SMILEScopy InChI
Affinity DataIC50: 282nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetCytoplasmic tyrosine-protein kinase BMX(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245603(CHEMBL4096207)copy SMILEScopy InChI
Affinity DataIC50: 341nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged BMX expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245615(CHEMBL4068683)copy SMILEScopy InChI
Affinity DataIC50: 365nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50161162(AVL-292 | CC-292 | Spebrutinib | US10596172, Compo...)copy SMILEScopy InChI
Affinity DataIC50: 442nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged wild-type EGFR (695 to end residues) expressed in baculovirus infected Sf9 insect cells using p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245598(CHEMBL4079595)copy SMILEScopy InChI
Affinity DataIC50: 596nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245601(CHEMBL4069186)copy SMILEScopy InChI
Affinity DataIC50: 667nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5HCKPubMed
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