Found 54 hits of Enzyme Inhibition Constant Data
TargetHistone deacetylase 5(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of human C-terminal His-tagged HDAC5 catalytic domain (656 to 1122 residues) expressed in baculovirus infected Sf9 insect cells using Boc-...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of human N-terminal GST-tagged HDAC7 (518 to end residues) expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substra...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 9(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human C-terminal His-tagged HDAC9 (604 to 1066 residues) expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substr...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of human N-terminal GST-tagged HDAC7 (518 to end residues) expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substra...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 9(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human C-terminal His-tagged HDAC9 (604 to 1066 residues) expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substr...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of human C-terminal His-tagged HDAC5 catalytic domain (656 to 1122 residues) expressed in baculovirus infected Sf9 insect cells using Boc-...More data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of human N-terminal GST-tagged HDAC7 (518 to end residues) expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substra...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 103nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 119nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 9(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human C-terminal His-tagged HDAC9 (604 to 1066 residues) expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substr...More data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of human C-terminal His-tagged HDAC5 catalytic domain (656 to 1122 residues) expressed in baculovirus infected Sf9 insect cells using Boc-...More data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of human C-terminal His-tagged HDAC5 catalytic domain (656 to 1122 residues) expressed in baculovirus infected Sf9 insect cells using Boc-...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 9(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Inhibition of human C-terminal His-tagged HDAC9 (604 to 1066 residues) expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substr...More data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Inhibition of human N-terminal GST-tagged HDAC7 (518 to end residues) expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substra...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of recombinant human HDAC6 expressed in HEK293 cells using Lys-Ac-AMC as substrate measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of recombinant human HDAC6 expressed in HEK293 cells using Lys-Ac-AMC as substrate measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of recombinant human HDAC6 expressed in HEK293 cells using Lys-Ac-AMC as substrate measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human full length C-terminal His-tagged HDAC8 expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substrate measure...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of human full length C-terminal His-tagged HDAC8 expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substrate measure...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]dofetilide from recombinant human ERG after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of recombinant human HDAC6 expressed in HEK293 cells using Lys-Ac-AMC as substrate measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 1.55E+4nMAssay Description:Inhibition of human full length C-terminal His-tagged HDAC8 expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substrate measure...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of HDAC6 in human A549 cells using tubulin as substrate measured after 4 hrs by Western blot analysisMore data for this Ligand-Target Pair
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of full length recombinant human C-terminal His-tagged HDAC3/N-terminal GST-tagged NCOR2 co-expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 2.58E+4nMAssay Description:Inhibition of full length recombinant human C-terminal His-tagged HDAC3/N-terminal GST-tagged NCOR2 co-expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
TargetHistone deacetylase 1/2/3/8(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of HDAC class 1 in human A549 cells using histone H4K12 as substrate measured after 4 hrs by Western blot analysisMore data for this Ligand-Target Pair
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 3.89E+4nMAssay Description:Inhibition of full length recombinant human C-terminal His-tagged HDAC3/N-terminal GST-tagged NCOR2 co-expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 3.97E+4nMAssay Description:Inhibition of human full length C-terminal FLAG/His-tagged HDAC1 expressed in baculovirus infected Sf9 insect cells using Lys-Ac-AMC as substrate mea...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of human full length C-terminal His-tagged HDAC8 expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substrate measure...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human full length C-terminal FLAG/His-tagged HDAC1 expressed in baculovirus infected Sf9 insect cells using Lys-Ac-AMC as substrate mea...More data for this Ligand-Target Pair
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of full length recombinant human C-terminal His-tagged HDAC3/N-terminal GST-tagged NCOR2 co-expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human full length C-terminal FLAG-tagged HDAC2 expressed in baculovirus infected Sf9 insect cells using Ac-Arg-Gly-Lys(Ac) as substrate...More data for this Ligand-Target Pair