Compile Data Set for Download or QSAR

Found 84 hits of Enzyme Inhibition Constant Data   

TargetNociceptin receptor(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529759(CHEMBL4451306)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-nociceptin from human nociceptin receptor expressed in cell membranes after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetNociceptin receptor(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529759(CHEMBL4451306)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-nociceptin from human nociceptin receptor expressed in cell membranes after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of SRC (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMedDrugBank
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of SRC (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMedDrugBank
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of Lyn B (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of Lyn B (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of CSK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of CSK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of Fyn A (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of Fyn A (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529757(CHEMBL4436086)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Inhibition of Lyn B (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529757(CHEMBL4436086)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Inhibition of Lyn B (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Inhibition of LCK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Inhibition of LCK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of BTK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of BTK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Inhibition of ABL1 (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Inhibition of ABL1 (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 5.30nMAssay Description:Inhibition of BRK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 5.30nMAssay Description:Inhibition of BRK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529755(CHEMBL4476482)copy SMILEScopy InChI
Affinity DataIC50: 182nMAssay Description:Inhibition of ABL1 (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529755(CHEMBL4476482)copy SMILEScopy InChI
Affinity DataIC50: 182nMAssay Description:Inhibition of ABL1 (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529755(CHEMBL4476482)copy SMILEScopy InChI
Affinity DataIC50: 191nMAssay Description:Inhibition of Fyn A (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529755(CHEMBL4476482)copy SMILEScopy InChI
Affinity DataIC50: 191nMAssay Description:Inhibition of Fyn A (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529755(CHEMBL4476482)copy SMILEScopy InChI
Affinity DataIC50: 209nMAssay Description:Inhibition of SRC (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529755(CHEMBL4476482)copy SMILEScopy InChI
Affinity DataIC50: 209nMAssay Description:Inhibition of SRC (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529755(CHEMBL4476482)copy SMILEScopy InChI
Affinity DataIC50: 237nMAssay Description:Inhibition of BTK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529755(CHEMBL4476482)copy SMILEScopy InChI
Affinity DataIC50: 237nMAssay Description:Inhibition of BTK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529757(CHEMBL4436086)copy SMILEScopy InChI
Affinity DataIC50: 287nMAssay Description:Inhibition of BTK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529757(CHEMBL4436086)copy SMILEScopy InChI
Affinity DataIC50: 287nMAssay Description:Inhibition of BTK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529757(CHEMBL4436086)copy SMILEScopy InChI
Affinity DataIC50: 402nMAssay Description:Inhibition of CSK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529757(CHEMBL4436086)copy SMILEScopy InChI
Affinity DataIC50: 402nMAssay Description:Inhibition of CSK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529755(CHEMBL4476482)copy SMILEScopy InChI
Affinity DataIC50: 442nMAssay Description:Inhibition of Lyn B (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529755(CHEMBL4476482)copy SMILEScopy InChI
Affinity DataIC50: 442nMAssay Description:Inhibition of Lyn B (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529756(CHEMBL1090672)copy SMILEScopy InChI
Affinity DataIC50: 456nMAssay Description:Inhibition of BTK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529756(CHEMBL1090672)copy SMILEScopy InChI
Affinity DataIC50: 456nMAssay Description:Inhibition of BTK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529758(CHEMBL4437669)copy SMILEScopy InChI
Affinity DataIC50: 473nMAssay Description:Inhibition of CSK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529758(CHEMBL4437669)copy SMILEScopy InChI
Affinity DataIC50: 473nMAssay Description:Inhibition of CSK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529756(CHEMBL1090672)copy SMILEScopy InChI
Affinity DataIC50: 478nMAssay Description:Inhibition of ABL1 (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529756(CHEMBL1090672)copy SMILEScopy InChI
Affinity DataIC50: 478nMAssay Description:Inhibition of ABL1 (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529755(CHEMBL4476482)copy SMILEScopy InChI
Affinity DataIC50: 515nMAssay Description:Inhibition of LCK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529755(CHEMBL4476482)copy SMILEScopy InChI
Affinity DataIC50: 515nMAssay Description:Inhibition of LCK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529758(CHEMBL4437669)copy SMILEScopy InChI
Affinity DataIC50: 626nMAssay Description:Inhibition of BRK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529758(CHEMBL4437669)copy SMILEScopy InChI
Affinity DataIC50: 626nMAssay Description:Inhibition of BRK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529756(CHEMBL1090672)copy SMILEScopy InChI
Affinity DataIC50: 626nMAssay Description:Inhibition of SRC (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529756(CHEMBL1090672)copy SMILEScopy InChI
Affinity DataIC50: 626nMAssay Description:Inhibition of SRC (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529758(CHEMBL4437669)copy SMILEScopy InChI
Affinity DataIC50: 644nMAssay Description:Inhibition of Lyn B (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529758(CHEMBL4437669)copy SMILEScopy InChI
Affinity DataIC50: 644nMAssay Description:Inhibition of Lyn B (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529756(CHEMBL1090672)copy SMILEScopy InChI
Affinity DataIC50: 704nMAssay Description:Inhibition of CSK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University of Silesia in Katowice

Curated by ChEMBL
LigandPNGBDBM50529756(CHEMBL1090672)copy SMILEScopy InChI
Affinity DataIC50: 704nMAssay Description:Inhibition of CSK (unknown origin) preincubated for 10 mins followed by substrate addition and measured after 1 hr by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P353VPubMed
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