Compile Data Set for Download or QSAR

Found 13 hits of Enzyme Inhibition Constant Data   

TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50523921(CHEMBL4446992)copy SMILEScopy InChI
Affinity DataIC50: 8.60nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92TPPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of c-MET (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92TPPubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50523921(CHEMBL4446992)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of VEGFR2 (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92TPPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50523921(CHEMBL4446992)copy SMILEScopy InChI
Affinity DataIC50: 352nMAssay Description:Inhibition of c-KIT (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92TPPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50523921(CHEMBL4446992)copy SMILEScopy InChI
Affinity DataIC50: 383nMAssay Description:Inhibition of c-SRC (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92TPPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50523921(CHEMBL4446992)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of EGFR (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92TPPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296349(CHEMBL4160329)copy SMILEScopy InChI
Affinity DataIC50: 3.35E+3nMAssay Description:Inhibition of c-MET (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92TPPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296396(CHEMBL4170935)copy SMILEScopy InChI
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of c-MET (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92TPPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50523925(CHEMBL4456688)copy SMILEScopy InChI
Affinity DataIC50: 4.24E+3nMAssay Description:Inhibition of c-MET (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92TPPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50523923(CHEMBL4456494)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of c-MET (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92TPPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50523922(CHEMBL4442035)copy SMILEScopy InChI
Affinity DataIC50: 4.52E+3nMAssay Description:Inhibition of c-MET (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92TPPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50523924(CHEMBL4445015)copy SMILEScopy InChI
Affinity DataIC50: 4.75E+3nMAssay Description:Inhibition of c-MET (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92TPPubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Zhuhai Campus of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50523921(CHEMBL4446992)copy SMILEScopy InChI
Affinity DataIC50: 6.66E+3nMAssay Description:Inhibition of IGF1R (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92TPPubMed
* indicates data uncertainty>20%