Compile Data Set for Download or QSAR

Found 166 hits of Enzyme Inhibition Constant Data   

TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50446130(AG-014699 | AG-14447 | RUCAPARIB CAMSYLATE | Rucap...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501829(CHEMBL4529965)copy SMILEScopy InChI
Affinity DataIC50: 0.646nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501829(CHEMBL4529965)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50446130(AG-014699 | AG-14447 | RUCAPARIB CAMSYLATE | Rucap...)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Inhibition of PARP1 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human full-length N-terminal GST-tagged PARP1 expressed in baculovirus infected Sf9 insect cells using histone as substrate measured af...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human full-length N-terminal GST-tagged PARP1 expressed in baculovirus infected Sf9 insect cells using histone as substrate measured af...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM27135(2-[(2R)-2-methylpyrrolidin-2-yl]-1H-1,3-benzodiazo...)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human full-length N-terminal GST-tagged PARP1 expressed in baculovirus infected Sf9 insect cells using histone as substrate measured af...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM27135(2-[(2R)-2-methylpyrrolidin-2-yl]-1H-1,3-benzodiazo...)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human full-length N-terminal GST-tagged PARP1 expressed in baculovirus infected Sf9 insect cells using histone as substrate measured af...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501836(CHEMBL4518901)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501836(CHEMBL4518901)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501827(CHEMBL4575227)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501827(CHEMBL4575227)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501835(CHEMBL4454914)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501830(CHEMBL4519178)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501830(CHEMBL4519178)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501835(CHEMBL4454914)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50188594(CHEBI:62878 | CHEMBL1086580)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human N-terminal GST-tagged TNKS2 (667 to 1166 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM27135(2-[(2R)-2-methylpyrrolidin-2-yl]-1H-1,3-benzodiazo...)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Inhibition of human PARP2 expressed in Escherichia coli using biotinylated histone H1 as substrate measured in presence of [3H]NAD+ by topcount scint...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501847(CHEMBL4446105)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501847(CHEMBL4446105)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501828(CHEMBL4586938)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501828(CHEMBL4586938)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501831(CHEMBL4450747)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501831(CHEMBL4450747)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501846(CHEMBL4539194)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501846(CHEMBL4539194)copy SMILEScopy InChI
Affinity DataIC50: 3.70nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501849(CHEMBL4469675)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501849(CHEMBL4469675)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501829(CHEMBL4529965)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Inhibition of human full-length N-terminal GST-tagged PARP1 expressed in baculovirus infected Sf9 insect cells using histone as substrate measured af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501829(CHEMBL4529965)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human full-length N-terminal GST-tagged PARP1 expressed in baculovirus infected Sf9 insect cells using histone as substrate measured af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501855(CHEMBL4474593)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501855(CHEMBL4474593)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50188594(CHEBI:62878 | CHEMBL1086580)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human N-terminal GST-tagged TNKS1 (1001 to 1327 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501848(CHEMBL4435102)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501848(CHEMBL4435102)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501832(CHEMBL4446923)copy SMILEScopy InChI
Affinity DataIC50: 4.80nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501832(CHEMBL4446923)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM27135(2-[(2R)-2-methylpyrrolidin-2-yl]-1H-1,3-benzodiazo...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human PARP1 expressed in Escherichia coli using biotinylated histone H1 as substrate measured in presence of [3H]NAD+ by topcount scint...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501829(CHEMBL4529965)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Inhibition of human N-terminal GST-tagged TNKS1 (1001 to 1327 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501829(CHEMBL4529965)copy SMILEScopy InChI
Affinity DataIC50: 8.80nMAssay Description:Inhibition of human N-terminal GST-tagged TNKS2 (667 to 1166 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501873(CHEMBL4515830)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501825(CHEMBL4576573)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501852(CHEMBL4471547)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501870(CHEMBL4458607)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501856(CHEMBL4583398)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501854(CHEMBL4437358)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501850(CHEMBL4470680)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50501844(CHEMBL4584942)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human N-terminal GST-tagged PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 insect cells using histone as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T156WFPubMed
Displayed 1 to 50 (of 166 total ) | Next | Last >>* indicates data uncertainty>20%