Compile Data Set for Download or QSAR

Found 4 hits of Enzyme Inhibition Constant Data   

TargetSerine/threonine-protein kinase 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50508990(CHEMBL4472294)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant full-length human MST1 assessed as residual activity using KKSRGDYMTMQIG as substrate measured after 40 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3PS5PubMed
TargetSerine/threonine-protein kinase 3(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50508990(CHEMBL4472294)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human MST2 (2 to end residues) assessed as residual activity using myelin basic protein as substrate measured after 40 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3PS5PubMed
TargetSerine/threonine-protein kinase LATS1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50508990(CHEMBL4472294)copy SMILEScopy InChI
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to recombinant human LATS1 (Q678 to V1130 residues) expressed in bacterial expression system assessed as dissociation constant by Ki...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3PS5PubMed
TargetSerine/threonine-protein kinase LATS2(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50508990(CHEMBL4472294)copy SMILEScopy InChI
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to wild-type human partial length LATS2 (Q641 to V1088 residues) expressed in mammalian expression system assessed as dissociation c...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3PS5PubMed
* indicates data uncertainty>20%