Compile Data Set for Download or QSAR

Found 314 hits of Enzyme Inhibition Constant Data   

LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against cytosolic c-SrcMore data for this Ligand-Target Pair
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of PI3K delta (unknown origin) by Adapta assayMore data for this Ligand-Target Pair
LigandPNGBDBM50537739(CHEMBL4648622 | US11230547, Compound 5-4)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537723(CHEMBL4639951 | US11230547, Compound 1-16)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537738(CHEMBL4633285 | US11230547, Compound 4-8)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537741(CHEMBL4637209 | US11179389, Compound 1-18)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibitory activity against cytosolic c-SrcMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537721(CHEMBL4646478 | US11230547, Compound 1-17)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:Inhibition of the fibroblast growth factor receptor (FGFR1)More data for this Ligand-Target Pair
LigandPNGBDBM50537737(CHEMBL4642953)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibition of the fibroblast growth factor receptor (FGFR1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537724(CHEMBL4643865 | US11230547, Compound 1-3)copy SMILEScopy InChI
Affinity DataIC50: 86nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537734(CHEMBL4642225 | US11230547, Compound 4-1)copy SMILEScopy InChI
Affinity DataIC50: 108nMAssay Description:Inhibitory activity against cytosolic c-SrcMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537725(CHEMBL4635168 | US11230547, Compound 2-1)copy SMILEScopy InChI
Affinity DataIC50: 161nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537732(CHEMBL4647402 | US11230547, Compound 3-3)copy SMILEScopy InChI
Affinity DataIC50: 165nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537740(CHEMBL4649678 | US11179389, Compound 1-13)copy SMILEScopy InChI
Affinity DataIC50: 185nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537738(CHEMBL4633285 | US11230547, Compound 4-8)copy SMILEScopy InChI
Affinity DataIC50: 187nMAssay Description:Inhibition of the fibroblast growth factor receptor (FGFR1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537741(CHEMBL4637209 | US11179389, Compound 1-18)copy SMILEScopy InChI
Affinity DataIC50: 219nMAssay Description:Inhibition of the fibroblast growth factor receptor (FGFR1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537725(CHEMBL4635168 | US11230547, Compound 2-1)copy SMILEScopy InChI
Affinity DataIC50: 258nMAssay Description:Inhibition of the fibroblast growth factor receptor (FGFR1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537733(CHEMBL4639546 | US11230547, Compound 4-2)copy SMILEScopy InChI
Affinity DataIC50: 263nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537734(CHEMBL4642225 | US11230547, Compound 4-1)copy SMILEScopy InChI
Affinity DataIC50: 329nMAssay Description:Inhibition of the fibroblast growth factor receptor (FGFR1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537719(CHEMBL4644618)copy SMILEScopy InChI
Affinity DataIC50: 364nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537735(CHEMBL4637750 | US11230547, Compound 4-3)copy SMILEScopy InChI
Affinity DataIC50: 374nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537743(CHEMBL4648691)copy SMILEScopy InChI
Affinity DataIC50: 474nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
LigandPNGBDBM50537737(CHEMBL4642953)copy SMILEScopy InChI
Affinity DataIC50: 557nMAssay Description:Inhibition of the fibroblast growth factor receptor (FGFR1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537740(CHEMBL4649678 | US11179389, Compound 1-13)copy SMILEScopy InChI
Affinity DataIC50: 737nMAssay Description:Inhibitory activity against cytosolic c-SrcMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537739(CHEMBL4648622 | US11230547, Compound 5-4)copy SMILEScopy InChI
Affinity DataIC50: 764nMAssay Description:Inhibitory activity against cytosolic c-SrcMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)copy SMILEScopy InChI
Affinity DataIC50: 884nMAssay Description:Inhibitory activity against cytosolic c-SrcMore data for this Ligand-Target Pair
LigandPNGBDBM50537722(CHEMBL4643688 | US11230547, Compound 1-18)copy SMILEScopy InChI
Affinity DataIC50: 918nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)copy SMILEScopy InChI
Affinity DataIC50: 945nMAssay Description:Inhibition of the fibroblast growth factor receptor (FGFR1)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537730(CHEMBL4649731 | US11230547, Compound 3-4)copy SMILEScopy InChI
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537736(CHEMBL4646437 | US11230547, Compound 4-4)copy SMILEScopy InChI
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537726(CHEMBL4635364 | US11230547, Compound 2-2)copy SMILEScopy InChI
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537727(CHEMBL4640850 | US11230547, Compound 2-3)copy SMILEScopy InChI
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537731(CHEMBL4640567 | US11230547, Compound 3-1)copy SMILEScopy InChI
Affinity DataIC50: 1.52E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537735(CHEMBL4637750 | US11230547, Compound 4-3)copy SMILEScopy InChI
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of the fibroblast growth factor receptor (FGFR1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537729(CHEMBL4644811 | US11230547, Compound 3-2)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537728(CHEMBL4646601 | US11230547, Compound 2-4)copy SMILEScopy InChI
Affinity DataIC50: 2.19E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537733(CHEMBL4639546 | US11230547, Compound 4-2)copy SMILEScopy InChI
Affinity DataIC50: 2.32E+3nMAssay Description:Inhibition of the fibroblast growth factor receptor (FGFR1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537723(CHEMBL4639951 | US11230547, Compound 1-16)copy SMILEScopy InChI
Affinity DataIC50: 2.96E+3nMAssay Description:Inhibitory activity against cytosolic c-SrcMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537726(CHEMBL4635364 | US11230547, Compound 2-2)copy SMILEScopy InChI
Affinity DataIC50: 4.12E+3nMAssay Description:Inhibition of the fibroblast growth factor receptor (FGFR1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)copy SMILEScopy InChI
Affinity DataIC50: 5.37E+3nMAssay Description:Inhibition of the fibroblast growth factor receptor (FGFR1)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537736(CHEMBL4646437 | US11230547, Compound 4-4)copy SMILEScopy InChI
Affinity DataIC50: 5.71E+3nMAssay Description:Inhibition of the fibroblast growth factor receptor (FGFR1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537727(CHEMBL4640850 | US11230547, Compound 2-3)copy SMILEScopy InChI
Affinity DataIC50: 6.97E+3nMAssay Description:Inhibitory activity against cytosolic c-SrcMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537720(CHEMBL4641286)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition Protein kinase C gammaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537721(CHEMBL4646478 | US11230547, Compound 1-17)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of the fibroblast growth factor receptor (FGFR1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537732(CHEMBL4647402 | US11230547, Compound 3-3)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of the fibroblast growth factor receptor (FGFR1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
LigandPNGBDBM50537724(CHEMBL4643865 | US11230547, Compound 1-3)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against cytosolic c-SrcMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)copy SMILEScopy InChI
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibitory activity against cytosolic c-SrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)copy SMILEScopy InChI
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibitory activity against cytosolic c-SrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of the fibroblast growth factor receptor (FGFR1)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
Displayed 1 to 50 (of 314 total ) | Next | Last >>* indicates data uncertainty>20%