Compile Data Set for Download or QSAR

Found 63 hits of Enzyme Inhibition Constant Data   

TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542172(CHEMBL4632760)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement [3H]ZM241385 from adenosine A2A receptor in human HeLa cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Displacement [3H]ZM241385 from adenosine A2A receptor in human HeLa cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542171(CHEMBL4645754)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement [3H]ZM241385 from adenosine A2A receptor in human HeLa cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542173(CHEMBL4634105)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement [3H]ZM241385 from adenosine A2A receptor in human HeLa cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50159488(CHEMBL3787197)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542194(CHEMBL4644677)copy SMILEScopy InChI
Affinity DataKi:  3.70nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542174(CHEMBL4632427)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Displacement [3H]ZM241385 from adenosine A2A receptor in human HeLa cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542190(CHEMBL4637285)copy SMILEScopy InChI
Affinity DataKi:  8.10nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542167(CHEMBL4645687)copy SMILEScopy InChI
Affinity DataKi:  8.30nMAssay Description:Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50159492(CHEMBL3786336)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50159486(CHEMBL3785290)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542166(CHEMBL4647965)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542168(CHEMBL4643113)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50159493(CHEMBL3785582)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542183(CHEMBL4637204)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50159497(CHEMBL3787034)copy SMILEScopy InChI
Affinity DataKi:  29nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542184(CHEMBL4644103)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50159499(CHEMBL3785618)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542178(CHEMBL4634269)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542191(CHEMBL4646279)copy SMILEScopy InChI
Affinity DataKi:  43nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542177(CHEMBL4641601)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)copy SMILEScopy InChI
Affinity DataKi:  66nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542193(CHEMBL4635502)copy SMILEScopy InChI
Affinity DataKi:  68nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)copy SMILEScopy InChI
Affinity DataKi:  73nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542166(CHEMBL4647965)copy SMILEScopy InChI
Affinity DataKi:  93nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542168(CHEMBL4643113)copy SMILEScopy InChI
Affinity DataKi:  99nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)copy SMILEScopy InChI
Affinity DataKi:  157nMAssay Description:Displacement [3H]ZM241385 from adenosine A2A receptor in human HeLa cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542188(CHEMBL4636018)copy SMILEScopy InChI
Affinity DataKi:  175nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542192(CHEMBL4636932)copy SMILEScopy InChI
Affinity DataKi:  215nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542169(CHEMBL4640980)copy SMILEScopy InChI
Affinity DataKi:  233nMAssay Description:Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542185(CHEMBL4643403)copy SMILEScopy InChI
Affinity DataKi:  278nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542169(CHEMBL4640980)copy SMILEScopy InChI
Affinity DataKi:  282nMAssay Description:Displacement [3H]ZM241385 from adenosine A2A receptor in human HeLa cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542170(CHEMBL4633188)copy SMILEScopy InChI
Affinity DataKi:  301nMAssay Description:Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542167(CHEMBL4645687)copy SMILEScopy InChI
Affinity DataKi:  340nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50159494(CHEMBL3785353)copy SMILEScopy InChI
Affinity DataKi:  371nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542173(CHEMBL4634105)copy SMILEScopy InChI
Affinity DataKi:  388nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542174(CHEMBL4632427)copy SMILEScopy InChI
Affinity DataKi:  402nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542169(CHEMBL4640980)copy SMILEScopy InChI
Affinity DataKi:  418nMAssay Description:Displacement [3H]NECA from adenosine A3 receptor in human HeLa cell membranes incubated for 180 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542175(CHEMBL4643705)copy SMILEScopy InChI
Affinity DataKi:  449nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50159495(CHEMBL3785635)copy SMILEScopy InChI
Affinity DataKi:  485nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542169(CHEMBL4640980)copy SMILEScopy InChI
Affinity DataKi:  508nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542176(CHEMBL4648862)copy SMILEScopy InChI
Affinity DataKi:  517nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)copy SMILEScopy InChI
Affinity DataKi:  683nMAssay Description:Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542181(CHEMBL4636116)copy SMILEScopy InChI
Affinity DataKi:  707nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542172(CHEMBL4632760)copy SMILEScopy InChI
Affinity DataKi:  708nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542186(CHEMBL4641123)copy SMILEScopy InChI
Affinity DataKi:  714nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542180(CHEMBL4644043)copy SMILEScopy InChI
Affinity DataKi:  721nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542189(CHEMBL4647365)copy SMILEScopy InChI
Affinity DataKi:  753nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50542171(CHEMBL4645754)copy SMILEScopy InChI
Affinity DataKi:  769nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD444SPubMed
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