Compile Data Set for Download or QSAR

Found 47 hits of Enzyme Inhibition Constant Data   

TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291482(2-[2-(2,4,6-Trimethyl-phenyl)-vinyl]-thiophene-3-s...)copy SMILEScopy InChI
Affinity DataIC50: 44nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291503(2-[2-(2,4,6-Trimethyl-phenyl)-ethyl]-thiophene-3-s...)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291490(3-[2-(2,4,6-Trimethyl-phenyl)-vinyl]-thiophene-2-s...)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291499(2-[2-(2,4-Dimethyl-phenyl)-ethyl]-thiophene-3-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291489(3-[2-(2,4,6-Trimethyl-phenyl)-ethyl]-thiophene-2-s...)copy SMILEScopy InChI
Affinity DataIC50: 58nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291486(2-[2-(6-Methyl-benzo[1,3]dioxol-5-yl)-ethyl]-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 62nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291491(3-[2-(6-Methyl-benzo[1,3]dioxol-5-yl)-vinyl]-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 72nMAssay Description:Tested for the inhibitory activity of cloned human ETA receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291498(3-{2-[6-(Tetrahydro-pyran-4-yloxymethyl)-benzo[1,3...)copy SMILEScopy InChI
Affinity DataIC50: 73nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291484(3-[2-(6-Hydroxymethyl-benzo[1,3]dioxol-5-yl)-vinyl...)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291488(2-[2-(6-Methyl-benzo[1,3]dioxol-5-yl)-vinyl]-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 81nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291500(3-[2-(6-Methyl-benzo[1,3]dioxol-5-yl)-ethyl]-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 91nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291496(3-[2-(2,4-Dimethyl-phenyl)-ethyl]-thiophene-2-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 102nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291501(2-(2-p-Tolyl-ethyl)-thiophene-3-sulfonic acid (4-b...)copy SMILEScopy InChI
Affinity DataIC50: 106nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291492(2-(2-Benzo[1,3]dioxol-5-yl-vinyl)-thiophene-3-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 141nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291483(2-[2-(2,4-Dimethyl-phenyl)-vinyl]-thiophene-3-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 166nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291495(3-[2-(2,4-Dimethyl-phenyl)-vinyl]-thiophene-2-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291485(2-(2-Benzo[1,3]dioxol-5-yl-ethyl)-thiophene-3-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 205nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291502(3-(2-Benzo[1,3]dioxol-5-yl-vinyl)-thiophene-2-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 218nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291493(2-(2-p-Tolyl-vinyl)-thiophene-3-sulfonic acid (4-b...)copy SMILEScopy InChI
Affinity DataIC50: 231nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291487(3-(2-Benzo[1,3]dioxol-5-yl-ethyl)-thiophene-2-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 237nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291494(3-(2-p-Tolyl-ethyl)-thiophene-2-sulfonic acid (4-b...)copy SMILEScopy InChI
Affinity DataIC50: 347nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50098772(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 630nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291497(3-(2-p-Tolyl-vinyl)-thiophene-2-sulfonic acid (4-b...)copy SMILEScopy InChI
Affinity DataIC50: 936nMAssay Description:Tested for its activity in cloned human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291489(3-[2-(2,4,6-Trimethyl-phenyl)-ethyl]-thiophene-2-s...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291490(3-[2-(2,4,6-Trimethyl-phenyl)-vinyl]-thiophene-2-s...)copy SMILEScopy InChI
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291482(2-[2-(2,4,6-Trimethyl-phenyl)-vinyl]-thiophene-3-s...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291503(2-[2-(2,4,6-Trimethyl-phenyl)-ethyl]-thiophene-3-s...)copy SMILEScopy InChI
Affinity DataIC50: 2.09E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291483(2-[2-(2,4-Dimethyl-phenyl)-vinyl]-thiophene-3-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 2.97E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291495(3-[2-(2,4-Dimethyl-phenyl)-vinyl]-thiophene-2-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 2.97E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291484(3-[2-(6-Hydroxymethyl-benzo[1,3]dioxol-5-yl)-vinyl...)copy SMILEScopy InChI
Affinity DataIC50: 3.24E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291488(2-[2-(6-Methyl-benzo[1,3]dioxol-5-yl)-vinyl]-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 3.28E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291499(2-[2-(2,4-Dimethyl-phenyl)-ethyl]-thiophene-3-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 3.48E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291493(2-(2-p-Tolyl-vinyl)-thiophene-3-sulfonic acid (4-b...)copy SMILEScopy InChI
Affinity DataIC50: 4.13E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291498(3-{2-[6-(Tetrahydro-pyran-4-yloxymethyl)-benzo[1,3...)copy SMILEScopy InChI
Affinity DataIC50: 4.14E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291496(3-[2-(2,4-Dimethyl-phenyl)-ethyl]-thiophene-2-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291492(2-(2-Benzo[1,3]dioxol-5-yl-vinyl)-thiophene-3-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 5.25E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291491(3-[2-(6-Methyl-benzo[1,3]dioxol-5-yl)-vinyl]-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 5.37E+3nMAssay Description:Tested for the inhibitory activity of cloned human ETB receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291497(3-(2-p-Tolyl-vinyl)-thiophene-2-sulfonic acid (4-b...)copy SMILEScopy InChI
Affinity DataIC50: 6.64E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291486(2-[2-(6-Methyl-benzo[1,3]dioxol-5-yl)-ethyl]-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289945(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291485(2-(2-Benzo[1,3]dioxol-5-yl-ethyl)-thiophene-3-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 9.24E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291494(3-(2-p-Tolyl-ethyl)-thiophene-2-sulfonic acid (4-b...)copy SMILEScopy InChI
Affinity DataIC50: 9.36E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291502(3-(2-Benzo[1,3]dioxol-5-yl-vinyl)-thiophene-2-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 9.96E+3nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291501(2-(2-p-Tolyl-ethyl)-thiophene-3-sulfonic acid (4-b...)copy SMILEScopy InChI
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291500(3-[2-(6-Methyl-benzo[1,3]dioxol-5-yl)-ethyl]-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291487(3-(2-Benzo[1,3]dioxol-5-yl-ethyl)-thiophene-2-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 1.79E+4nMAssay Description:Inhibition of human Endothelin B receptor using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291481(2-(2,4,6-Trimethyl-phenoxymethyl)-thiophene-3-sulf...)copy SMILEScopy InChI
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibitory of human Endothelin A receptor by using I-ET-1 as radioligand in a competitive radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HKC
* indicates data uncertainty>20%