Compile Data Set for Download or QSAR

Found 583 hits of Enzyme Inhibition Constant Data   

TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 0.403nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225517(GTC000226A | GTC000226B)copy SMILEScopy InChI
Affinity DataIC50: 0.412nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225517(GTC000226A | GTC000226B)copy SMILEScopy InChI
Affinity DataIC50: 0.746nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225519(GTC000227A)copy SMILEScopy InChI
Affinity DataIC50: 0.75nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225519(GTC000227A)copy SMILEScopy InChI
Affinity DataIC50: 0.857nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 0.869nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225517(GTC000226A | GTC000226B)copy SMILEScopy InChI
Affinity DataIC50: 0.925nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 0.977nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225520(GTC000228A | GTC000228B | GTC000228C)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225523(GTC000229A)copy SMILEScopy InChI
Affinity DataIC50: 1.19nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.26nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.27nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225562(GTC000266A | GTC000266B | GTC000266C)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225520(GTC000228A | GTC000228B | GTC000228C)copy SMILEScopy InChI
Affinity DataIC50: 1.38nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225523(GTC000229A)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225525(GTC000231A)copy SMILEScopy InChI
Affinity DataIC50: 1.42nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.43nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225524(GTC000230A)copy SMILEScopy InChI
Affinity DataIC50: 1.46nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225520(GTC000228A | GTC000228B | GTC000228C)copy SMILEScopy InChI
Affinity DataIC50: 1.47nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225530(GTC000236A)copy SMILEScopy InChI
Affinity DataIC50: 1.48nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.48nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.51nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.54nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.56nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225538(GTC000242A)copy SMILEScopy InChI
Affinity DataIC50: 1.58nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.61nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.61nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.61nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.62nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225529(GTC000235A)copy SMILEScopy InChI
Affinity DataIC50: 1.64nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.66nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.66nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.75nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.83nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225531(GTC000237A | GTC000237B)copy SMILEScopy InChI
Affinity DataIC50: 1.87nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225528(GTC000234A)copy SMILEScopy InChI
Affinity DataIC50: 1.87nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.91nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.91nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.92nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.92nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 1.93nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225529(GTC000235A)copy SMILEScopy InChI
Affinity DataIC50: 1.94nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225545(GTC000249A)copy SMILEScopy InChI
Affinity DataIC50: 1.99nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225520(GTC000228A | GTC000228B | GTC000228C)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 2.01nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 2.01nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225527(GTC000233A)copy SMILEScopy InChI
Affinity DataIC50: 2.02nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase SYK [355-635](Homo sapiens (Human))
D3R

LigandPNGBDBM225520(GTC000228A | GTC000228B | GTC000228C)copy SMILEScopy InChI
Affinity DataIC50: 2.02nMAssay Description:SYK assay_HTRFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GM1PubMed
Displayed 1 to 50 (of 583 total ) | Next | Last >>* indicates data uncertainty>20%