Found 92 hits of Enzyme Inhibition Constant Data
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 103nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 125nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 133nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 138nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 153nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 183nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 197nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 243nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 413nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 433nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 553nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 760nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.05E+3nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.53E+3nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 2.15E+3nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to the NK2 receptor assayed by displacement of [125I]-Neurokinin AMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to the NK2 receptor assayed by displacement of [125I]-Neurokinin AMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to the NK2 receptor assayed by displacement of [125I]-Neurokinin AMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to the NK2 receptor assayed by displacement of [125I]-Neurokinin AMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to the NK2 receptor assayed by displacement of [125I]-Neurokinin AMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to the NK2 receptor assayed by displacement of [125I]-Neurokinin AMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to the NK2 receptor assayed by displacement of [125I]-Neurokinin AMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to the NK2 receptor assayed by displacement of [125I]-Neurokinin AMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair