Compile Data Set for Download or QSAR

Found 7 hits of Enzyme Inhibition Constant Data   

TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50469862(CHEMBL409219)copy SMILEScopy InChI
Affinity DataKi:  0.0135nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BW7PubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50469858(CHEMBL268397)copy SMILEScopy InChI
Affinity DataKi:  0.0234nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BW7PubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50469859(A-75998 | CHEMBL263839)copy SMILEScopy InChI
Affinity DataKi:  0.0316nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BW7PubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50469856(CHEMBL263840 | ORG-30850)copy SMILEScopy InChI
Affinity DataKi:  0.0331nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BW7PubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50469857(CHEMBL268319)copy SMILEScopy InChI
Affinity DataKi:  0.0525nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BW7PubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50469860(CHEMBL409990)copy SMILEScopy InChI
Affinity DataKi:  0.0617nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BW7PubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50469861(CHEMBL438829)copy SMILEScopy InChI
Affinity DataKi:  0.117nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BW7PubMed
* indicates data uncertainty>20%