Affinity Data by PubMed id=8759641

Found 48 hits of Enzyme Inhibition Constant Data

Glutamate receptor ionotropic, NMDA 2C(Rattus norvegicus (Rat))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM17662((2S)-2-amino-3-(3-hydroxy-5-methyl-1,2-oxazol-4-yl...)copy SMILEScopy InChI

IC50: 1.00E+5nMAssay Description:The compound was evaluated for agonist to competitive inhibition of radioligand ([3H]- CPP ) at Ionotropic Excitatory Amino acid receptorsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052554(2-Amino-6-(3-hydroxy-5-methyl-isoxazol-4-yl)-hexan...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM85356((S)-2-Aminoadipic acid | CAS_542-32-5)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50004852(AMAA | Amino-(3-hydroxy-5-methyl-isoxazol-4-yl)-ac...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonist activityof the compound at Metabotropic Excitatory Amino acid Receptors Expressed in CHO cells. mGlu2More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 4(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052555(2-Amino-5-(3-hydroxy-5-methyl-isoxazol-4-yl)-penta...)copy SMILEScopy InChI

EC50: >3.00E+6nMAssay Description:Agonistic activity at mGlu4a receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052555(2-Amino-5-(3-hydroxy-5-methyl-isoxazol-4-yl)-penta...)copy SMILEScopy InChI

EC50: 4.10E+5nMAssay Description:Agonistic activity at mGlu6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052552(2-Amino-octanedioic acid | CHEMBL320957)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 4(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052553((2S)-2-aminohexanedioic acid | (S)-2-aminohexanedi...)copy SMILEScopy InChI

EC50: >3.00E+6nMAssay Description:Agonistic activity at mGlu4a receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052553((2S)-2-aminohexanedioic acid | (S)-2-aminohexanedi...)copy SMILEScopy InChI

EC50: 1.40E+5nMAssay Description:Agonistic activity at mGlu6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052552(2-Amino-octanedioic acid | CHEMBL320957)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 1(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM17662((2S)-2-amino-3-(3-hydroxy-5-methyl-1,2-oxazol-4-yl...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonist activityof the compound at Metabotropic Excitatory Amino acid Receptors Expressed in CHO cells. mGlu1-alphaMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 1(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50026947((R)-2-Amino-3-(3-hydroxy-5-methyl-isoxazol-4-yl)-p...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonist activityof the compound at Metabotropic Excitatory Amino acid Receptors Expressed in CHO cells. mGlu1-alphaMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM17662((2S)-2-amino-3-(3-hydroxy-5-methyl-1,2-oxazol-4-yl...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonist activityof the compound at Metabotropic Excitatory Amino acid Receptors Expressed in CHO cells. mGlu2More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 1(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052551(2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-butyr...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu1-alpha receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 4(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)copy SMILEScopy InChI

EC50: 1.50E+4nMAssay Description:Agonistic activity at mGlu4a receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052555(2-Amino-5-(3-hydroxy-5-methyl-isoxazol-4-yl)-penta...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 1(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM31174(CHEMBL29757 | D-Aspartate | D-Aspartic Acid)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu1-alpha receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50026947((R)-2-Amino-3-(3-hydroxy-5-methyl-isoxazol-4-yl)-p...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonist activityof the compound at Metabotropic Excitatory Amino acid Receptors Expressed in CHO cells. mGlu6More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)copy SMILEScopy InChI

EC50: 8.50E+3nMAssay Description:Agonistic activity at mGlu2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 1(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052552(2-Amino-octanedioic acid | CHEMBL320957)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu1-alpha receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 1(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50004852(AMAA | Amino-(3-hydroxy-5-methyl-isoxazol-4-yl)-ac...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonist activityof the compound at Metabotropic Excitatory Amino acid Receptors Expressed in CHO cells. mGlu1-alphaMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052551(2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-butyr...)copy SMILEScopy InChI

EC50: 8.20E+4nMAssay Description:Agonistic activity at mGlu6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
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Details Article
BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 1(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)copy SMILEScopy InChI

EC50: 1.90E+4nMAssay Description:Agonistic activity at mGlu1-alpha receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50026947((R)-2-Amino-3-(3-hydroxy-5-methyl-isoxazol-4-yl)-p...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonist activityof the compound at Metabotropic Excitatory Amino acid Receptors Expressed in CHO cells. mGlu2More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 1(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052553((2S)-2-aminohexanedioic acid | (S)-2-aminohexanedi...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu1-alpha receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052554(2-Amino-6-(3-hydroxy-5-methyl-isoxazol-4-yl)-hexan...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM17662((2S)-2-amino-3-(3-hydroxy-5-methyl-1,2-oxazol-4-yl...)copy SMILEScopy InChI

EC50: 2.20E+5nMAssay Description:Agonist activityof the compound at Metabotropic Excitatory Amino acid Receptors Expressed in CHO cells. mGlu6More data for this Ligand-Target Pair

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Details Article
BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM31174(CHEMBL29757 | D-Aspartate | D-Aspartic Acid)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM85356((S)-2-Aminoadipic acid | CAS_542-32-5)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052551(2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-butyr...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 1(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM85356((S)-2-Aminoadipic acid | CAS_542-32-5)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu1-alpha receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052549(2-Amino-heptanedioic acid | CHEMBL111050)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 1(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052555(2-Amino-5-(3-hydroxy-5-methyl-isoxazol-4-yl)-penta...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu1-alpha receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052549(2-Amino-heptanedioic acid | CHEMBL111050)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 4(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052551(2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-butyr...)copy SMILEScopy InChI

EC50: >3.00E+6nMAssay Description:Agonistic activity at mGlu4a receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052553((2S)-2-aminohexanedioic acid | (S)-2-aminohexanedi...)copy SMILEScopy InChI

EC50: 3.50E+4nMAssay Description:Agonistic activity at mGlu2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 4(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM17662((2S)-2-amino-3-(3-hydroxy-5-methyl-1,2-oxazol-4-yl...)copy SMILEScopy InChI

EC50: >3.00E+6nMAssay Description:Agonist activityof the compound at Metabotropic Excitatory Amino acid Receptors Expressed in CHO cells. mGlu4aMore data for this Ligand-Target Pair

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Details Article
BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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Details Article
BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)copy SMILEScopy InChI

EC50: 2.00E+4nMAssay Description:Agonistic activity at mGlu6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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Details Article
BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM31174(CHEMBL29757 | D-Aspartate | D-Aspartic Acid)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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Details Article
BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 1(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu1-alpha receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 1(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052554(2-Amino-6-(3-hydroxy-5-methyl-isoxazol-4-yl)-hexan...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu1-alpha receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 1(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50052549(2-Amino-heptanedioic acid | CHEMBL111050)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu1-alpha receptor expressed in CHO cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM50004852(AMAA | Amino-(3-hydroxy-5-methyl-isoxazol-4-yl)-ac...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonist activityof the compound at Metabotropic Excitatory Amino acid Receptors Expressed in CHO cells. mGlu6More data for this Ligand-Target Pair

Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

Metabotropic glutamate receptor 1(Homo sapiens (Human))
Royal Danish School of Pharmacy

Curated by ChEMBL

BDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)copy SMILEScopy InChI

EC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu1-alpha receptor expressed in CHO cellsMore data for this Ligand-Target Pair

PDB
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Details Article
BindingDB Entry DOI: 10.7270/Q2M909BHPubMed

* indicates data uncertainty>20%