Compile Data Set for Download or QSAR

Found 92 hits of Enzyme Inhibition Constant Data   

TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058111(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058080(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058106(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058114(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058105(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058099(Acetic acid 2-(6-{[3-(4-chloro-3-methyl-isoxazol-5...)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058117(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 5.10nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058097(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 5.60nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058103(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058075(Acetic acid 2-(6-{[3-(4-chloro-3-methyl-isoxazol-5...)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058084(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 6.60nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058092(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 6.80nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058077(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 9.30nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058115(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058116(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 10.8nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058093(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058100(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058108(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058095(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058109(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058086(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058104(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058072(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058096(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058102(3-(3,4-Dimethyl-isoxazol-5-ylsulfamoyl)-thiophene-...)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058081(3-(3,4-Dimethyl-isoxazol-5-ylsulfamoyl)-thiophene-...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058112(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058091(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058076(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058089(3-{[3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-th...)copy SMILEScopy InChI
Affinity DataIC50: 62nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058101(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058107(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058083(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 104nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058113(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 132nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058078(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 146nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058073(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 166nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058110(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058088(2-{[3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-th...)copy SMILEScopy InChI
Affinity DataIC50: 214nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058090(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 229nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058074(2-{[3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-t...)copy SMILEScopy InChI
Affinity DataIC50: 549nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058094(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 838nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058085(2-[(3-Methoxy-phenylamino)-methyl]-thiophene-3-sul...)copy SMILEScopy InChI
Affinity DataIC50: 933nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058079(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 977nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058098(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)copy SMILEScopy InChI
Affinity DataIC50: 1.29E+3nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058087(2-{[3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-t...)copy SMILEScopy InChI
Affinity DataIC50: 1.43E+3nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058082(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 1.91E+3nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin A receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058104(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 4.37E+3nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin B receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058091(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 5.89E+3nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin B receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058110(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 6.17E+3nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin B receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
ImmunoPharmaceutics Inc.

Curated by ChEMBL
LigandPNGBDBM50058112(3-(4-Bromo-3-methyl-isoxazol-5-ylsulfamoyl)-thioph...)copy SMILEScopy InChI
Affinity DataIC50: 6.92E+3nMAssay Description:In vitro inhibition of endothelin binding to human Endothelin B receptor using [125I]-labeled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3JKTPubMed
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