Reaction Details
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Target
Protein-glutamine gamma-glutamyltransferase 6
Ligand
BDBM577483
Substrate
n/a
Meas. Tech.
Transamidation Assay for Determining Inhibitor Selectivity
IC50
17.0±n/a nM
Citation
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More Info.:
Target
Name:
Protein-glutamine gamma-glutamyltransferase 6
Synonyms:
Protein-glutamine gamma-glutamyltransferase 6 | TG6 | TGM3L | TGM3L_HUMAN | TGM6 | TGY | TGase Y | TGase-3-like | TGase-6 | Transglutaminase Y | Transglutaminase-3-like | Transglutaminase-6 | Transglutaminase-6 (TG6)
Type:
Protein
Mol. Mass.:
79319.01
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
706
Sequence:
MAGIRVTKVDWQRSRNGAAHHTQEYPCPELVVRRGQSFSLTLELSRALDCEEILIFTMETGPRASEALHTKAVFQTSELERGEGWTAAREAQMEKTLTVSLASPPSAVIGRYLLSIRLSSHRKHSNRRLGEFVLLFNPWCAEDDVFLASEEERQEYVLSDSGIIFRGVEKHIRAQGWNYGQFEEDILNICLSILDRSPGHQNNPATDVSCRHNPIYVTRVISAMVNSNNDRGVVQGQWQGKYGGGTSPLHWRGSVAILQKWLKGRYKPVKYGQCWVFAGVLCTVLRCLGIATRVVSNFNSAHDTDQNLSVDKYVDSFGRTLEDLTEDSMWNFHVWNESWFARQDLGPSYNGWQVLDATPQEESEGVFRCGPASVTAIREGDVHLAHDGPFVFAEVNADYITWLWHEDESRERVYSNTKKIGRCISTKAVGSDSRVDITDLYKYPEGSRKERQVYSKAVNRLFGVEASGRRIWIRRAGGRCLWRDDLLEPATKPSIAGKFKVLEPPMLGHDLRLALCLANLTSRAQRVRVNLSGATILYTRKPVAEILHESHAVRLGPQEEKRIPITISYSKYKEDLTEDKKILLAAMCLVTKGEKLLVEKDITLEDFITIKVLGPAMVGVAVTVEVTVVNPLIERVKDCALMVEGSGLLQEQLSIDVPTLEPQERASVQFDITPSKSGPRQLQVDLVSPHFPDIKGFVIVHVATAK