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Target
AGAP001281-PB
Ligand
BDBM600747
Substrate
n/a
Meas. Tech.
thallium-flux assay
IC50
12100±n/a nM
Citation
 Swale, DR; Foil, LD Method for controlling hematophagous or sap-feeding arthropods US Patent  US11632953 Publication Date 4/25/2023
Target
Name:
AGAP001281-PB
Synonyms:
n/a
Type:
Protein
Mol. Mass.:
49315.66
Organism:
African malaria mosquito
Description:
A7UVQ1
Residue:
426
Sequence:
MAAERPTLDEKKPLNRIFMRPGVIEEEPDSLDSVISNLPLTVVPSLARISTHGSAFSRQESVRSRALRPGTTRKYRRRAILKNGDCNIVLSKVSRQRLRFLQDIFTTLVDAQWRWTLLVFAFSFIGSWLFFGAIWWLIAFTHGDLEEMHLPKNQEESGWKPCVFNIESYTSAFLFSIETQTTIGYGYRTTTEECPEAIFIMCFQSIYGVMMQAFMVGFVFAKMTRPKHRTQTLLFSKHAVVCQRDGELSLMFRVGDMRKSHIIGANIRAQLIRTKLSREGEVMAQYQHELEVGADHCGSDLFFIWPQIVTHRINTESPFYNMSASDLLQDRFEIVVILEGTVESTGQSTQARSSYVNTEILWGHRFEPIVFYNKENQVYEINYSKFNETHSVDTPLCSARELAEFYKYQDDYRNQAEDHHHLQTPA
  
Inhibitor
Name:
BDBM600747
Synonyms:
US11632953, Compound 4 | VU0650729
Type:
Small organic molecule
Emp. Form.:
C19H20N2O2
Mol. Mass.:
308.3743
SMILES:
O=C(Cn1ccc2c1CCCC2=O)N1CCCc2ccccc12
Structure:
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