Reaction Details
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Target
GTPase KRas [G12C,C51S,C80L,C118S]
Ligand
BDBM625378
Substrate
n/a
Meas. Tech.
Biochemical Functional Assay
IC50
29.0±n/a nM
Citation
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More Info.:
Target
Name:
GTPase KRas [G12C,C51S,C80L,C118S]
Synonyms:
GTPase KRas (1-169)(G12C)(C51S)(C80L)(C118S)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
19417.19
Organism:
Homo sapiens (Human)
Description:
P01116[G12C,C51S,C80L,C118S]
Residue:
169
Sequence:
MTEYKLVVVGACGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETSLLDILDTAGQEEYSAMRDQYMRTGEGFLLVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKSDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQRVEDAFYTLVREIRQYRLK