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Target
Cathepsin G
Ligand
BDBM37097
Substrate
n/a
Meas. Tech.
Cathepsin G dose-response confirmation
IC50
631.087±41.0064 nM
Citation
 PubChem, PC Cathepsin G dose-response confirmation PubChem Bioassay (2008)[AID]
Target
Name:
Cathepsin G
Synonyms:
CATG_HUMAN | CG | CTSG
Type:
PROTEIN
Mol. Mass.:
28860.08
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469016
Residue:
255
Sequence:
MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSFKLLDQMETPL
  
Inhibitor
Name:
BDBM37097
Synonyms:
MLS000087437 | N-cyclohexyl-7-methoxy-4,5-dihydrobenz[g]indoxazene-3-carboxamide | N-cyclohexyl-7-methoxy-4,5-dihydrobenzo[g][1,2]benzoxazole-3-carboxamide | N-cyclohexyl-7-methoxy-4,5-dihydronaphtho[2,1-d]isoxazole-3-carboxamide | SMR000023660 | cid_3245662
Type:
Small organic molecule
Emp. Form.:
C19H22N2O3
Mol. Mass.:
326.3896
SMILES:
COc1ccc2-c3onc(C(=O)NC4CCCCC4)c3CCc2c1
Structure:
Search PDB for entries with ligand similarity: