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Target
Cathepsin G
Ligand
BDBM32791
Substrate
n/a
Meas. Tech.
Cathepsin G dose-response confirmation
IC50
4328.64±215.521 nM
Citation
 PubChem, PC Cathepsin G dose-response confirmation PubChem Bioassay (2008)[AID]
Target
Name:
Cathepsin G
Synonyms:
CATG_HUMAN | CG | CTSG
Type:
PROTEIN
Mol. Mass.:
28860.08
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469016
Residue:
255
Sequence:
MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSFKLLDQMETPL
  
Inhibitor
Name:
BDBM32791
Synonyms:
1-(1-benzothien-3-ylcarbonyl)-1H-pyrazole | 1-benzothiophen-3-yl(1-pyrazolyl)methanone | 1-benzothiophen-3-yl(pyrazol-1-yl)methanone | MLS000065687 | SMR000080341 | benzothiophen-3-yl(pyrazol-1-yl)methanone | cid_841465
Type:
Small organic molecule
Emp. Form.:
C12H8N2OS
Mol. Mass.:
228.27
SMILES:
O=C(c1csc2ccccc12)n1cccn1
Structure:
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