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Target
Cathepsin G
Ligand
BDBM32794
Substrate
n/a
Meas. Tech.
Cathepsin G dose-response confirmation
IC50
10754.1±788.726 nM
Citation
 PubChem, PC Cathepsin G dose-response confirmation PubChem Bioassay (2008)[AID]
Target
Name:
Cathepsin G
Synonyms:
CATG_HUMAN | CG | CTSG
Type:
PROTEIN
Mol. Mass.:
28860.08
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469016
Residue:
255
Sequence:
MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSFKLLDQMETPL
  
Inhibitor
Name:
BDBM32794
Synonyms:
1-benzoyl-3,6,6-trimethyl-1,5,6,7-tetrahydro-4H-indazol-4-one | 1-benzoyl-3,6,6-trimethyl-5,7-dihydroindazol-4-one | 3,6,6-trimethyl-1-(phenylcarbonyl)-5,7-dihydroindazol-4-one | MLS000060946 | SMR000069174 | cid_749826
Type:
Small organic molecule
Emp. Form.:
C17H18N2O2
Mol. Mass.:
282.337
SMILES:
Cc1nn(C(=O)c2ccccc2)c2CC(C)(C)CC(=O)c12
Structure:
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