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Target
Beta-2 adrenergic receptor
Ligand
BDBM50036835
Substrate
n/a
Ki
100±n/a nM
Comments
PDSP_659
Citation
 Bylund, DB; Snyder, SH Beta adrenergic receptor binding in membrane preparations from mammalian brain. Mol Pharmacol 12:568-80 (1976) [PubMed]
Target
Name:
Beta-2 adrenergic receptor
Synonyms:
ADRB2 | ADRB2R | ADRB2_HUMAN | B2AR | Beta-2 adrenoceptor | Beta-2 adrenoreceptor
Type:
n/a
Mol. Mass.:
46461.69
Organism:
Homo sapiens (Human)
Description:
P07550
Residue:
413
Sequence:
MGQPGNGSAFLLAPNGSHAPDHDVTQERDEVWVVGMGIVMSLIVLAIVFGNVLVITAIAKFERLQTVTNYFITSLACADLVMGLAVVPFGAAHILMKMWTFGNFWCEFWTSIDVLCVTASIETLCVIAVDRYFAITSPFKYQSLLTKNKARVIILMVWIVSGLTSFLPIQMHWYRATHQEAINCYANETCCDFFTNQAYAIASSIVSFYVPLVIMVFVYSRVFQEAKRQLQKIDKSEGRFHVQNLSQVEQDGRTGHGLRRSSKFCLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIQDNLIRKEVYILLNWIGYVNSGFNPLIYCRSPDFRIAFQELLCLRRSSLKAYGNGYSSNGNTGEQSGYHVEQEKENKLLCEDLPGTEDFVGHQGTVPSDNIDSQGRNCSTNDSLL
  
Inhibitor
Name:
BDBM50036835
Synonyms:
1-(3,4-Dichloro-phenyl)-2-isopropylamino-ethanol | 1-(3,4-Dichloro-phenyl)-2-isopropylamino-ethanol(Di chloroisoproterenol) | CHEMBL30816 | Dichloroisoproterenol,(+/-)
Type:
Small organic molecule
Emp. Form.:
C11H15Cl2NO
Mol. Mass.:
248.149
SMILES:
CC(C)NCC(O)c1ccc(Cl)c(Cl)c1
Structure:
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