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Target
Muscarinic acetylcholine receptor M4
Ligand
BDBM81799
Substrate
n/a
Ki
100±n/a nM
Comments
PDSP_932
Citation
 Waelbroeck, M; Tastenoy, M; Camus, J; Christophe, J Binding of selective antagonists to four muscarinic receptors (M1 to M4) in rat forebrain. Mol Pharmacol 38:267-73 (1990) [PubMed]
Target
Name:
Muscarinic acetylcholine receptor M4
Synonyms:
ACM4_MOUSE | Cholinergic, muscarinic M4 | Chrm-4 | Chrm4 | Mm4 mAChR | Muscarinic acetylcholine receptor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
53004.88
Organism:
MOUSE
Description:
Cholinergic, muscarinic M4 CHRM4 MOUSE::P32211
Residue:
479
Sequence:
MANFTPVNGSSANQSVRLVTTAHNHLETVEMVFIATVTGSLSLVTVVGNILVMLSIKVNRQLQTVNNYFLFSLACADLIIGAFSMNLYTLYIIKGYWPLGAVVCDLWLALDYVVSNASVMNLLIISFDRYFCVTKPLTYPARRTTKMAGLMIAAAWVLSFVLWAPAILFWQFVVGKRTVPDNQCFIQFLSNPAVTFGTAIAAFYLPVVIMTVLYIHISLASRSRVHKHRPEGPKEKKAKTLAFLKSPLMKPSIKKPPPGGASREELRNGKLEEAPPPALPPPPRPVADKDTSNESSSGSATQNTKERPPTELSTTEAATTPALPAPTLQPRTLNPASKWSKIQIVTKQTGSECVTAIEIVPATPAGMRPAANVARKFASIARNQVRKKRQMAARERKVTRTIFAILLAFILTWTPYNVMVLVNTFCQSCIPERVWSIGYWLCYVNSTINPACYALCNATFKKTFRHLLLCQYRNIGTAR
  
Inhibitor
Name:
BDBM81799
Synonyms:
CAS_98299-40-2 | HHSiD | NSC_3602 | hexahydrosiladifenidol
Type:
Small organic molecule
Emp. Form.:
C20H33NOSi
Mol. Mass.:
331.5676
SMILES:
O[Si](CCCN1CCCCC1)(C1CCCCC1)c1ccccc1
Structure:
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